Atazanavir

Atazanavir

SCHEMBL29362158

COC(=O)N[C@H](C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CN(Cc1ccc(-c2ccccn2)cc1)NC(=O)[C@@H](NC(=O)OC)C(C)(C)C)C(C)(C)C.O=S(=O)(O)O

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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The experimentally established mechanism targets of Atazanavir. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT1A1 P22309 3/20 0.94
MLNR O43193 1/20 0.94
NR1I2 O75469 1/20 0.94
SLCO2B1 O94956 1/20 0.94
ABCB11 O95342 1/20 0.94
ABCB1 P08183 1/20 0.94
CCKAR P32238 1/20 0.94
OPRK1 P41145 1/20 0.94
GHSR Q92847 1/20 0.94
SLCO1B3 Q9NPD5 1/20 0.94
ABCG2 Q9UNQ0 1/20 0.94
SLCO1B1 Q9Y6L6 1/20 0.94
KCNH2 Q12809 1/20 0.69
CTSD P07339 4/20 0.55
CYP3A4 P08684 3/20 0.55
CTSE P14091 1/20 0.39
PGC P20142 1/20 0.39
PSEN1 P49768 8/20 0.38
PSEN2 P49810 8/20 0.38
APH1B Q8WW43 8/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Atazanavir SCHEMBL27785902 1.00 UGT1A1 (0.94) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Atazanavir SCHEMBL341700 1.00 UGT1A1 (0.94) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Atazanavir SCHEMBL291519 1.00 UGT1A1 (0.94) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Atazanavir SCHEMBL28121836 1.00 UGT1A1 (0.94) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Atazanavir SCHEMBL22847477 0.97 UGT1A1 (1.00) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Atazanavir SCHEMBL21565117 0.97 UGT1A1 (1.00) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Atazanavir SCHEMBL20629937 0.97 UGT1A1 (1.00) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Atazanavir SCHEMBL20629941 0.97 UGT1A1 (1.00) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Atazanavir SCHEMBL825777 0.97 UGT1A1 (1.00) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Atazanavir SCHEMBL7993264 0.97 UGT1A1 (1.00) UGT1A1MLNRNR1I2SLCO2B1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 157 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12459989-B2 Antibody therapies for human immunodeficiency virus (HIV) BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2025-11-04 US claimed
US-20250170172-A1 METHODS FOR TREATING LENTIVIRUS INFECTION JERICHO SCIENCES LLC (US) 2025-05-29 US claimed
EP-4394098-A1 PREPARATION METHOD FOR COLLAGEN FIBER, COLLAGEN FIBER, AND USE Zhejiang Heuristic New Material Technology Limited Liability Company (CN) 2024-07-03 EP claimed
EP-3960735-B1 QUINAZOLINE DERIVATIVES USED TO TREAT HIV GILEAD SCIENCES INC (US) 2023-09-13 EP claimed
WO-2023164293-A1 METHODS FOR VIRAL INFECTIONS JERICHO SCIENCES, LLC (US) 2023-08-31 WO claimed
US-20230000884-A1 COMBINATION THERAPY FOR TREATING COVID-19 Luckwel Pharmaceuticals Inc. 2023-01-05 US claimed
EP-3656384-B1 COMBINATIONS COMPRISING 5-PHENOXY-3H-PYRIMIDIN-4-ONE DERIVATIVES AND THEIR USE FOR THE PROPHYLAXIS OR TREATMENT OF INFECTION BY HIV MERCK SHARP & DOHME (US) 2022-02-23 EP claimed
US-20220025021-A1 ANTIBODY THERAPIES FOR HUMAN IMMUNODEFICIENCY VIRUS (HIV) BETH ISRAEL DEACONESS MEDICAL CENTER, INC. 2022-01-27 US claimed
US-20260132139-A1 HIV INHIBITOR COMPOUNDS GILEAD SCIENCES INC (US) 2026-05-14 US disclosed
US-12617843-B2 Human broadly neutralizing antibodies against the membrane-proximal external region of HIV Env for vaccine design and intervention THE SCRIPPS RESEARCH INSTITUTE (US) 2026-05-05 US disclosed
WO-2026085583-A1 MOLECULAR ASSAY FOR DETECTING HIV-1 DRUG-RESISTANT MUTATIONS ST VINCENT'S HOSPITAL SYDNEY LIMITED (AU) 2026-04-30 WO disclosed
EP-4731212-A1 COMBINATION THERAPIES OF FASN INHIBITORS WITH THYROID HORMONE RECEPTOR AGONISTS Sagimet Biosciences Inc. (US) 2026-04-29 EP disclosed
EP-4730340-A1 METHOD FOR DETERMINING THE PRESENCE OF A PROBE SEQUENCE IN A TARGET NUCLEOTIDE SEQUENCE Institut Pasteur de Dakar (SN) 2026-04-22 EP disclosed
US-20260102464-A1 METHODS AND COMPOSITIONS FOR PREVENTING AND TREATING ATHEROSCLEROSIS AND RELATED DISEASES SHANGHAI PUYOU BIOMEDICAL CO LTD (CN) 2026-04-16 US disclosed
EP-3974831-A1 METHODS FOR DETECTING THE PRESENCE OF A BACTERIUM IN A WHOLE BLOOD SAMPLE T2 Biosystems, Inc. (US) 2022-03-30 EP disclosed
US-20220062293-A1 MODULATORS OF TOLL-LIKE RECEPTORS FOR THE TREATMENT OF HIV GILEAD SCIENCES, INC. 2022-03-03 US disclosed
CN-114081867-A Method for improving drug loading capacity of microspheres 中国药科大学 2022-02-25 CN disclosed
WO-2022040435-A1 NANODRUGS FOR TARGETED DRUG DELIVERY AND USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-02-24 WO disclosed
EP-3955921-A1 2-IMINO-5-OXO-IMIDAZOLIDINE INHIBITORS OF HIV PROTEASE GILEAD SCIENCES, INC. (US) 2022-02-23 EP disclosed
US-20220025021-A1 ANTIBODY THERAPIES FOR HUMAN IMMUNODEFICIENCY VIRUS (HIV) BETH ISRAEL DEACONESS MEDICAL CENTER, INC. 2022-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250170172-A1 METHODS FOR TREATING LENTIVIRUS INFECTION ZC3HAV1, ZC3HAV1L, ZFR UGT1A1 3785/4885MLNR 4368/4885NR1I2 3306/4885
US-12617843-B2 Human broadly neutralizing antibodies against the membrane-proximal external region of HIV Env for vaccine design and intervention CD4, VSIG8, IGLV6-57 UGT1A1 4033/4885MLNR 4497/4885NR1I2 3805/4885
US-20260102464-A1 METHODS AND COMPOSITIONS FOR PREVENTING AND TREATING ATHEROSCLEROSIS AND RELATED DISEASES APOL1, APOB, LDLR UGT1A1 4523/4885MLNR 4808/4885NR1I2 1886/4885
US-20260132139-A1 HIV INHIBITOR COMPOUNDS SLC11A2, SLC6A15, NHERF1 UGT1A1 1885/4885MLNR 3606/4885NR1I2 2239/4885
US-20220062293-A1 MODULATORS OF TOLL-LIKE RECEPTORS FOR THE TREATMENT OF HIV TLR7, TLR3, TLR6 UGT1A1 923/4885MLNR 181/4885NR1I2 417/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.