SCHEMBL29382265

SCHEMBL29382265

COc1cc(COC(=O)CCCC/C=C/C(C)C)ccc1O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 13/20 0.68
CYP1A2 P05177 4/20 0.68
CYP3A4 P08684 4/20 0.68
CYP2D6 P10635 3/20 0.68
ALDH1A1 P00352 2/20 0.68
ALOX5 P09917 2/20 0.68
CYP2C9 P11712 2/20 0.68
CYP2C19 P33261 2/20 0.68
MEN1 O00255 2/20 0.68
MAPT P10636 2/20 0.68
KMT2A Q03164 2/20 0.68
TP53 P04637 2/20 0.68
KDM1A O60341 1/20 0.68
NR1I2 O75469 1/20 0.68
LMNA P02545 1/20 0.68
ADORA3 P0DMS8 1/20 0.68
ALOX15 P16050 1/20 0.68
PTGS1 P23219 1/20 0.68
HTR2C P28335 1/20 0.68
MAPK1 P28482 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1585964 1.00 TRPV1 (0.68) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL15358922 0.91 TRPV1 (0.58) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL14329163 0.87 TRPV1 (0.53) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL5923227 0.86 TRPV1 (0.73) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL20036237 0.86 TRPV1 (0.62) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL5923219 0.86 TRPV1 (0.73) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL2210228 0.86 LTA4H (0.53) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL14092947 0.86 ALDH1A1 (0.54) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL6002616 0.86 ALDH1A1 (0.54) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL16407907 0.85 TRPV1 (0.54) TRPV1CYP1A2CYP3A4CYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 154 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4210687-B1 TRPV1 AGONISTS IN THE PREVENTION OF DIABETIC ULCERS IMPERIAL COLLEGE INNOVATIONS LTD (GB) 2026-05-27 EP claimed
EP-4739298-A1 ACTIVATORS OF THE XC- SYSTEM AND/OR GPX-4 FOR TREATING CONDITIONS ASSOCIATED WITH CONE PHOTORECEPTOR DEGENERATION SORBONNE UNIVERSITE (FR) 2026-05-13 EP claimed
US-20260047592-A1 NUTRITIONAL SUPPLEMENT COMPOSITION AND RELATED MANUFACTURING PROCESS CHEN YUHUA (US) 2026-02-19 US claimed
EP-4680210-A1 MEDICAL PATCH COMPRISING SKIN IRRITATING ACTIVE AGENT LTS Lohmann Therapie-Systeme AG (DE) 2026-01-21 EP claimed
US-12274680-B2 Treatment of benign prostatic hypertrophy with capsinoids CREASY II GEORGE WILLIAM (US) 2025-04-15 US claimed
WO-2025012137-A1 ACTIVATORS OF THE XC- SYSTEM AND/OR GPX-4 FOR TREATING CONDITIONS ASSOCIATED WITH CONE PHOTORECEPTOR DEGENERATION SORBONNE UNIVERSITE (FR) 2025-01-16 WO claimed
WO-2025012667-A1 ACTIVATORS OF THE XC-SYSTEM AND/OR GPX-4 FOR TREATING CONDITIONS ASSOCIATED WITH CONE PHOTORECEPTOR DEGENERATION. SORBONNE UNIVERSITE (FR) 2025-01-16 WO claimed
US-20250017251-A1 DIETARY SUPPLEMENT CONTAINING CAYENNE PEPPER POWDER PERFECT SPORTS INC (CA) 2025-01-16 US claimed
US-12109268-B2 Nanoparticle delivery system for targeted anti-obesity treatment UNIVERSITY OF WYOMING (US) 2024-10-08 US claimed
WO-2024189213-A1 MEDICAL PATCH COMPRISING SKIN IRRITATING ACTIVE AGENT LTS LOHMANN THERAPIE-SYSTEME AG (DE) 2024-09-19 WO claimed
US-20230012268-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INFLAMMATION WITH STEROIDS AND A MODULATOR BUZZELET DEVELOPMENT AND TECHNOLOGIES LTD (IL) 2023-01-12 US claimed
EP-4114372-A1 USE OF QX314 TO PREVENT SYMPATHOEXCITATION ASSOCIATED WITH ADMINISTRATION OF TRPV1 MODULATORS Neucures, Inc. (US) 2023-01-11 EP claimed
EP-4072558-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INFLAMMATION WITH STEROIDS AND A MODULATOR Buzzelet Development And Technologies Ltd (IL) 2022-10-19 EP claimed
WO-2022182940-A1 NEURAL CONTROL OF ADAPTIVE IMMUNITY THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2022-09-01 WO claimed
US-20220233463-A1 LOCAL ANESTHETIC COMPRISING A TRP CHANNEL MODULATOR BUZZELET DEVELOPMENT AND TECHNOLOGIES LTD (IL) 2022-07-28 US claimed
EP-4017486-A1 COMPOSITONS FOR THE TREATMENT OF A CONDITION CHARACTERIZED BY ANANDAMIDE DEFICIENCY AND USES THEREOF Buzzelet Development And Technologies Ltd (IL) 2022-06-29 EP claimed
US-20220168246-A1 COMPOSITONS FOR THE TREATMENT OF A CONDITION CHARACTERIZED BY ANANDAMIDE DEFICIENCY AND USES THEREOF BUZZELET DEVELOPMENT AND TECHNOLOGIES LTD (IL) 2022-06-02 US claimed
WO-2022079574-A1 COMPOSITIONS FOR REDUCING INFLAMMATION TO IMPROVE OR MAINTAIN MENTAL OR PHYSICAL HEALTH GOODCAP PHARMACEUTICALS LTD. (CA) 2022-04-21 WO claimed
WO-2022063372-A1 ORAL ANTAGONIST COMPOSITIONS FOR NICOTINE BURNING RELIEF FERTIN PHARMA A/S (DK) 2022-03-31 WO claimed
EP-3968970-A1 LOCAL ANESTHETIC COMPRISING A TRP CHANNEL MODULATOR Buzzelet Development And Technologies Ltd (IL) 2022-03-23 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260047592-A1 NUTRITIONAL SUPPLEMENT COMPOSITION AND RELATED MANUFACTURING PROCESS CHIA, COL2A1, COL1A1 TRPV1 502/4885CYP1A2 2390/4885CYP3A4 3400/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.