Perphenazine

Perphenazine

SCHEMBL29385591

OCCN1CCN(CCCN2c3ccccc3Sc3ccc(Cl)cc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2

The experimentally established mechanism targets of Perphenazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 6/20 1.00
MAPT P10636 8/20 1.00
LMNA P02545 8/20 1.00
MAPK1 P28482 7/20 1.00
CYP2D6 P10635 7/20 1.00
CYP3A4 P08684 6/20 1.00
SMN1; SMN2 Q16637 6/20 1.00
ADRA2A P08913 6/20 1.00
ADRA2B P18089 6/20 1.00
ADRA2C P18825 6/20 1.00
SLC6A2 P23975 6/20 1.00
HTR2A P28223 6/20 1.00
SLC6A4 P31645 6/20 1.00
HRH1 P35367 6/20 1.00
DRD3 P35462 6/20 1.00
HTR2B P41595 6/20 1.00
NPSR1 Q6W5P4 5/20 1.00
TP53 P04637 5/20 1.00
ABCB11 O95342 5/20 1.00
HTR1A P08908 5/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Perphenazine SCHEMBL8762197 1.00 MAPT (1.00) MAPTLMNAMAPK1CYP2D6CYP3A4
Perphenazine SCHEMBL29461866 1.00 MAPT (1.00) MAPTLMNAMAPK1CYP2D6CYP3A4
Perphenazine SCHEMBL42125 1.00 MAPT (1.00) MAPTLMNAMAPK1CYP2D6CYP3A4
Perphenazine SCHEMBL140891 0.99 MAPT (0.98) MAPTLMNAMAPK1CYP2D6CYP3A4
Perphenazine SCHEMBL145754 0.99 MAPT (0.98) MAPTLMNAMAPK1CYP2D6CYP3A4
Perphenazine SCHEMBL29846305 0.99 MAPT (0.98) MAPTLMNAMAPK1CYP2D6CYP3A4
Perphenazine SCHEMBL5307579 0.96 MAPT (0.91) MAPTLMNAMAPK1CYP2D6CYP3A4
Perphenazine SCHEMBL28086447 0.96 MAPT (0.91) MAPTLMNAMAPK1CYP2D6CYP3A4
Perphenazine SCHEMBL28456705 0.94 MAPT (0.88) MAPTLMNAMAPK1CYP2D6CYP3A4
Perphenazine SCHEMBL8014634 0.94 MAPT (0.88) MAPTLMNAMAPK1CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 87 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748885-A1 POLYCARBONATE COMPOSITIONS HAVING IMPROVED TRANSMITTANCE AND DUCTILITY PROPERTIES SHPP Global Technologies B.V. (NL) 2026-05-27 EP claimed
US-20250084247-A1 Polycarbonate Compositions with Flame Retardant Properties for Laser Activating Plating Processes SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2025-03-13 US claimed
EP-4444797-A1 POLYCARBONATE COMPOSITIONS WITH FLAME RETARDANT PROPERTIES FOR LASER ACTIVATING PLATING PROCESSES SHPP Global Technologies B.V. (NL) 2024-10-16 EP claimed
CN-118525059-A Polycarbonate compositions with flame retardant properties for laser activated plating processes 高新特殊工程塑料全球技术有限公司 2024-08-20 CN claimed
WO-2023131915-A1 POLYCARBONATE COMPOSITIONS WITH FLAME RETARDANT PROPERTIES FOR LASER ACTIVATING PLATING PROCESSES SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2023-07-13 WO claimed
EP-4209553-A1 POLYCARBONATE COMPOSITIONS WITH FLAME RETARDANT PROPERTIES FOR LASER ACTIVATING PLATING PROCESSES SHPP Global Technologies B.V. (NL) 2023-07-12 EP claimed
US-11649357-B2 Laser platable thermoplastic compositions with good flame retardancy, high heat property and good ductility and shaped articles made therefrom SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2023-05-16 US claimed
US-20220062291-A1 COMPOSITIONS AND METHODS OF TREATING CANCERS BY ADMINISTERING A PHENOTHIAZINE-RELATED DRUG THAT ACTIVATES PROTEIN PHOSPHATASE 2A (PP2A) WITH REDUCED INHIBITORY ACTIVITY TARGETED TO THE DOPAMINE D2 RECEPTOR AND ACCOMPANYING TOXICITY DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-03-03 US claimed
EP-4748885-A1 POLYCARBONATE COMPOSITIONS HAVING IMPROVED TRANSMITTANCE AND DUCTILITY PROPERTIES SHPP Global Technologies B.V. (NL) 2026-05-27 EP disclosed
WO-2026099586-A1 DRY POWDER FORMULATIONS NANOPHARM LIMITED (GB) 2026-05-15 WO disclosed
US-12569486-B2 Calmodulin inhibitors, CHK2 inhibitors and RSK inhibitors for the treatment of ribosomal disorders and ribosomapathies THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2026-03-10 US disclosed
US-12565563-B2 Halogen-free synergist AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2026-03-03 US disclosed
EP-4690102-A1 METHOD AND COMPOSITIONS FOR ANALYZING TOXICITY IN ORGANISMS vivoVerse, LLC (US) 2026-02-11 EP disclosed
US-12523664-B2 Sensor chip and methods thereof NATIONAL UNIVERSITY OF SINGAPORE (SG) 2026-01-13 US disclosed
WO-2022094615-A1 COMPOUNDS AND METHODS FOR INCREASED ANTISENSE ACTIVITY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-05-05 WO disclosed
WO-2022055285-A1 PHARMACEUTICAL COMPOSITION FOR KILLING CANCER PROGENITOR CELLS 연세대학교 산학협력단 2022-03-17 WO disclosed
CN-107750177-B Use of antistatic materials in airways for hot aerosol condensation processes 艾利斯达医药品公司 2022-03-11 CN disclosed
US-20220062291-A1 COMPOSITIONS AND METHODS OF TREATING CANCERS BY ADMINISTERING A PHENOTHIAZINE-RELATED DRUG THAT ACTIVATES PROTEIN PHOSPHATASE 2A (PP2A) WITH REDUCED INHIBITORY ACTIVITY TARGETED TO THE DOPAMINE D2 RECEPTOR AND ACCOMPANYING TOXICITY DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-03-03 US disclosed
US-20220062291-A1 COMPOSITIONS AND METHODS OF TREATING CANCERS BY ADMINISTERING A PHENOTHIAZINE-RELATED DRUG THAT ACTIVATES PROTEIN PHOSPHATASE 2A (PP2A) WITH REDUCED INHIBITORY ACTIVITY TARGETED TO THE DOPAMINE D2 RECEPTOR AND ACCOMPANYING TOXICITY DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-03-03 US disclosed
CN-114042074-A Combined medication method for synergistically treating human brain glioma 东南大学 2022-02-15 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12569486-B2 Calmodulin inhibitors, CHK2 inhibitors and RSK inhibitors for the treatment of ribosomal disorders and ribosomapathies RPS6KA1, RPS6KA2, RPS6KA3 DRD2 3909/4885MAPT 2118/4885LMNA 1109/4885
US-20220062291-A1 COMPOSITIONS AND METHODS OF TREATING CANCERS BY ADMINISTERING A PHENOTHIAZINE-RELATED DRUG THAT ACTIVATES PROTEIN PHOSPHATASE 2A (PP2A) WITH REDUCED INHIBITORY ACTIVITY TARGETED TO THE DOPAMINE D2 RECEPTOR AND ACCOMPANYING TOXICITY PPP2CA, PPP2R2A, PPP3CA DRD2 619/4885MAPT 2082/4885LMNA 4630/4885
US-12565563-B2 Halogen-free synergist PPOX, PFAS, DUOX2 DRD2 2172/4885MAPT 952/4885LMNA 4272/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.