Setiptiline

Setiptiline

SCHEMBL29396748

CN1CCC2=C(C1)c1ccccc1Cc1ccccc12.O=C(O)/C=C\C(=O)O

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Setiptiline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 known ✓ P21728 7/20 0.76
ADRA2A known ✓ P08913 2/20 0.76
HTR1A known ✓ P08908 1/20 0.76
SLC6A2 known ✓ P23975 1/20 0.76
SLC6A4 known ✓ P31645 1/20 0.76
ADRA1A known ✓ P35348 1/20 0.76
SLC6A3 known ✓ Q01959 1/20 0.76
DRD2 known ✓ P14416 6/20 0.50
ADRA2B known ✓ P18089 1/20 0.50
HTR2A known ✓ P28223 1/20 0.50
HTR2C known ✓ P28335 1/20 0.50
HRH1 known ✓ P35367 1/20 0.50
DRD3 P35462 6/20 0.76
CHRM2 P08172 2/20 0.76
CHRM1 P11229 2/20 0.76
OPRM1 P35372 1/20 0.76
KCNH2 Q12809 1/20 0.76
CYP3A4 P08684 2/20 0.51
HTT P42858 1/20 0.51
DRD5 P21918 6/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Setiptiline SCHEMBL623015 1.00 DRD1 (0.76) DRD1DRD3CHRM2ADRA2ACHRM1
Setiptiline SCHEMBL29414110 0.87 DRD1 (1.00) DRD1DRD3CHRM2ADRA2ACHRM1
Setiptiline SCHEMBL211362 0.87 DRD1 (1.00) DRD1DRD3CHRM2ADRA2ACHRM1
Maleic Acid SCHEMBL167958 0.81 DRD2 (0.59) DRD1DRD3CHRM2ADRA2ACHRM1
Fumaric Acid SCHEMBL12467794 0.81 DRD2 (0.59) DRD1DRD3CHRM2ADRA2ACHRM1
SCHEMBL10728179 0.81 DRD1 (0.86) DRD1DRD3CHRM2ADRA2ACHRM1
SCHEMBL10730066 0.77 DRD1 (0.69) DRD1DRD3CHRM2ADRA2ACHRM1
Maleic Acid SCHEMBL11488022 0.75 CYP3A4 (0.50) DRD1DRD3CHRM2ADRA2ACHRM1
Fumaric Acid SCHEMBL11488028 0.75 CYP3A4 (0.50) DRD1DRD3CHRM2ADRA2ACHRM1
SCHEMBL12355565 0.73 DRD1 (0.73) DRD1DRD3CHRM2ADRA2ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115223082-B Aerial video classification method based on space-time multi-scale convertors 重庆邮电大学 2025-06-10 CN disclosed
CN-119229319-B Aerial video classification model and method 重庆市地理信息和遥感应用中心(重庆市测绘产品质量检验测试中心) 2025-05-30 CN disclosed
CN-119229319-A Local semantic enhancement encoder, window semantic enhancement transducer block, aerial video classification model and method 重庆市地理信息和遥感应用中心(重庆市测绘产品质量检验测试中心) 2024-12-31 CN disclosed
WO-2024093624-A1 MEASUREMENT METHOD AND APPARATUS, AND TERMINAL AND NETWORK DEVICE 大唐移动通信设备有限公司 2024-05-10 WO disclosed
US-11916820-B2 Reference signal configuration, information transmission, and information receiving methods and device ZTE CORPORATION (CN) 2024-02-27 US disclosed
CN-117542118-A Unmanned aerial vehicle aerial video action recognition method based on space-time information dynamic modeling 中国科学技术大学 2024-02-09 CN disclosed
CN-113573286-B Method and apparatus for performing device-to-device communication between user devices SK电信有限公司 2024-01-05 CN disclosed
CN-116614885-A Communication method, device, terminal, network equipment and storage medium 中国移动通信有限公司研究院 2023-08-18 CN disclosed
CN-108111280-B Reference signal configuration, information transmission and information receiving method and device 中兴通讯股份有限公司 2023-07-14 CN disclosed
US-20230198699-A1 REFERENCE SIGNAL CONFIGURATION, INFORMATION TRANSMISSION, AND INFORMATION RECEIVING METHODS AND DEVICE ZTE CORPORATION (CN) 2023-06-22 US disclosed
EP-3595232-B1 Apparatus and method for transmitting/receiving downlink data channel signal transmission information in cellular radio communication system using cooperative multi-point scheme SAMSUNG ELECTRONICS CO LTD (KR) 2023-04-26 EP disclosed
CN-114637031-B Beidou civil dual-frequency satellite-based enhanced message communication method and device 中国人民解放军32021部队 2023-02-28 CN disclosed
CN-115223082-A Aerial video classification method based on space-time multi-scale transform 重庆邮电大学 2022-10-21 CN disclosed
CN-112020144-B Method and equipment for determining resources of asynchronous physical uplink shared channel 华为技术有限公司 2022-09-02 CN disclosed
CN-114637031-A Beidou civil dual-frequency satellite-based enhanced message communication method and device 中国人民解放军32021部队 2022-06-17 CN disclosed
US-11337037-B2 Multicast service reading and sending method, and related device HUAWEI TECHNOLOGIES CO., LTD (CN) 2022-05-17 US disclosed
CN-109272033-B Online soft interval kernel learning algorithm based on step length control 中国石油大学(华东) 2022-03-08 CN disclosed