SCHEMBL29401039

SCHEMBL29401039

NCc1cc(F)cc(C(N)=O)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.47
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
MAOB P27338 2/20 0.41
PARP10 Q53GL7 2/20 0.41
PLAU P00749 1/20 0.37
LOXL2 Q9Y4K0 3/20 0.37
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
KCNH2 Q12809 1/20 0.36
PTPN11 Q06124 1/20 0.36
MAPK8 P45983 1/20 0.36
HCAR1 Q9BXC0 1/20 0.35
CYP3A4 P08684 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22501583 1.00 PARP1 (0.47) PARP1CES2CES1MAOBPARP10
SCHEMBL31469843 0.85 PLAU (0.42) PARP1PARP10PLAULOXL2CYP3A4
SCHEMBL4613289 0.85 PLAU (0.42) PARP1PARP10PLAULOXL2CYP3A4
SCHEMBL16951666 0.84 CYP4F2 (0.47) PARP1CES2CES1MAOBPARP10
SCHEMBL15888156 0.84 HCAR1 (0.53) CES2CES1LOXL2HCAR1
SCHEMBL9970966 0.82 PARP1 (0.46) PARP1CES2CES1MAOBPARP10
SCHEMBL7077548 0.80 PARP1 (0.60) PARP1CES2CES1PTPN11HCAR1
SCHEMBL259315 0.80 CES2 (0.62) PARP1CES2CES1PTPN11HCAR1
SCHEMBL27824440 0.79 CES2 (0.38) CES2CES1LOXL2HCAR1SMN1; SMN2
SCHEMBL3874944 0.78 LOXL2 (0.58) LOXL2PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114127050-A Benzopyran and imidazole derivatives useful for stabilizing amyloidogenic immunoglobulin light chains 斯克利普斯研究所 2022-03-01 CN disclosed