SCHEMBL29407693

SCHEMBL29407693

C[Si](C)(C)CCOCn1ccc2c(N)ncnc21

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 4/20 0.40
WDR77 Q9BQA1 4/20 0.40
ADK P55263 1/20 0.38
ENPP1 P22413 2/20 0.35
DGAT1 O75907 1/20 0.35
PI4KA P42356 1/20 0.35
PI4K2B Q8TCG2 1/20 0.35
PI4K2A Q9BTU6 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
NT5E P21589 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13738818 1.00 PRMT5 (0.40) PRMT5WDR77ADKENPP1DGAT1
SCHEMBL13243594 0.85 DGAT1 (0.38) PRMT5WDR77DGAT1
SCHEMBL18547536 0.84 DGAT1 (0.40) DGAT1
SCHEMBL98891 0.84 FGFR1 (0.35) DGAT1
SCHEMBL127257 0.84 DGAT1 (0.35) DGAT1
SCHEMBL6672255 0.83 USP2 (0.40) PRMT5WDR77ADKENPP1
SCHEMBL13737015 0.83 XDH (0.39) PRMT5WDR77DGAT1
SCHEMBL20893945 0.83 ALDH1A1 (0.36) PRMT5WDR77DGAT1
SCHEMBL17858713 0.82 DGAT1 (0.30) DGAT1
SCHEMBL29416267 0.82 DGAT1 (0.30) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119874707-A FGFR inhibitors and methods of use thereof 传达治疗有限公司 2025-04-25 CN disclosed
CN-114126620-B FGFR inhibitors and methods of use thereof 传达治疗有限公司 2024-12-31 CN disclosed
EP-4424311-A2 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS Cystic Fibrosis Foundation (US) 2024-09-04 EP disclosed
EP-3541390-B1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUND (US) 2024-05-01 EP disclosed
CN-117425660-A Aromatic heterocyclic compound, intermediate thereof, pharmaceutical composition and application 上海翊石医药科技有限公司 2024-01-19 CN disclosed
CN-114126620-A FGFR inhibitors and methods of use thereof 传达治疗有限公司 2022-03-01 CN disclosed