SCHEMBL29419554

SCHEMBL29419554

CCOC(=O)Cc1cc2cccnc2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
RIPK1 Q13546 5/20 0.45
HSD17B10 Q99714 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TP53 P04637 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
DAO P14920 1/20 0.44
MAPT P10636 2/20 0.42
HRH4 Q9H3N8 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CHEK1 O14757 1/20 0.41
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
RECQL P46063 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29587495 0.80 DAO (0.51) RIPK1DAOHRH4HRH3
SCHEMBL29602065 0.79 RIPK1 (0.51) RIPK1DAOHRH4HRH3
SCHEMBL29588892 0.79 RIPK1 (0.52) RIPK1DAOHRH4HRH3
SCHEMBL30568660 0.78 HSD17B10 (0.54) SMN1; SMN2HSD17B10KDM4EALDH1A1TP53
SCHEMBL832252 0.78 KDM4E (0.58) SMN1; SMN2RIPK1HSD17B10KDM4EALDH1A1
SCHEMBL170083 0.77 HSD17B10 (0.56) SMN1; SMN2HSD17B10KDM4EALDH1A1HPGD
SCHEMBL1939638 0.76 DRD2 (0.50) RIPK1DAOMAPT
SCHEMBL3380080 0.76 HSD17B10 (0.65) SMN1; SMN2HSD17B10KDM4EALDH1A1TP53
SCHEMBL29765495 0.75 RIPK1 (0.44) RIPK1DAOHRH4HRH3
SCHEMBL253780 0.75 ALDH1A1 (0.54) RIPK1KDM4EALDH1A1HTTDAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110724142-B Amide or sulfonamide substituted hydrazine derivatives as JAK kinase inhibitors 启元生物(杭州)有限公司 2022-09-02 CN disclosed
CN-114685505-A Imidazopyrrolopyridines as JAK family kinase inhibitors 詹森药业有限公司 2022-07-01 CN disclosed
CN-114478528-A Aroyl-substituted tricyclic compound, preparation method and application thereof 劲方医药科技(上海)有限公司 2022-05-13 CN disclosed
CN-110312719-B Imidazopyrrolopyridines as JAK family kinase inhibitors 詹森药业有限公司 2022-04-15 CN disclosed
CN-110088105-B Small molecule inhibitors of JAK family kinases 詹森药业有限公司 2022-03-18 CN disclosed