SCHEMBL29587495

SCHEMBL29587495

O=C(O)Cc1cc2cccnc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.51
RIPK1 Q13546 11/20 0.47
DRD2 P14416 2/20 0.46
DRD4 P21917 2/20 0.46
DRD3 P35462 2/20 0.46
CCNE1 P24864 1/20 0.45
CDK2 P24941 1/20 0.45
HRH4 Q9H3N8 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29588892 0.86 RIPK1 (0.52) DAORIPK1DRD2DRD4DRD3
SCHEMBL1100944 0.84 DAO (0.49) DAORIPK1DRD2DRD4DRD3
SCHEMBL29602065 0.83 RIPK1 (0.51) DAORIPK1DRD2DRD4DRD3
SCHEMBL27151128 0.81 DAO (0.49) DAORIPK1DRD2DRD4DRD3
SCHEMBL5677159 0.80 DAO (0.59) DAORIPK1HRH4HRH3
SCHEMBL29419554 0.80 SMN1; SMN2 (0.49) DAORIPK1HRH4HRH3
SCHEMBL13543890 0.80 RIPK1 (0.58) DAORIPK1DRD2DRD4DRD3
SCHEMBL29765495 0.79 RIPK1 (0.44) DAORIPK1DRD2DRD4DRD3
SCHEMBL18361821 0.77 RIPK1 (0.48) DAORIPK1DRD2DRD4DRD3
SCHEMBL29460523 0.77 RIPK1 (0.60) DAORIPK1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685505-A Imidazopyrrolopyridines as JAK family kinase inhibitors 詹森药业有限公司 2022-07-01 CN disclosed
CN-114478528-A Aroyl-substituted tricyclic compound, preparation method and application thereof 劲方医药科技(上海)有限公司 2022-05-13 CN disclosed