SCHEMBL29423933

SCHEMBL29423933

CCOC(=O)[C@@]1(CC)[C@@H]2Cc3cc(OCc4ccc(C)c(Br)c4)ccc3[C@H]21

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 10/20 0.41
ADAM17 P78536 2/20 0.36
HPD P32754 1/20 0.35
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
ALOX5 P09917 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29423931 0.85 FFAR1 (0.36) FFAR1ADAM17ALOX5
SCHEMBL29423946 0.80 CDK8 (0.37) FFAR1
SCHEMBL29423937 0.75 FFAR1 (0.34) FFAR1
SCHEMBL18940289 0.74 FFAR1 (0.48) FFAR1HPDMRGPRX4
SCHEMBL18632583 0.69 NPC1 (0.41) FFAR1MRGPRX4
SCHEMBL29423909 0.65 MAOB (0.47) FFAR1MAOAMAOBMRGPRX4
SCHEMBL18632561 0.65 SHBG (0.40) NPSR1
SCHEMBL24650797 0.62 CHRNB2 (0.43) FFAR1
SCHEMBL7038455 0.61 GAA (0.56) NPSR1
SCHEMBL4611333 0.61 HPGD (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3974413-A1 ANTIDIABETIC SUBSTITUTED HETEROARYL COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2022-03-30 EP disclosed