SCHEMBL29439748

SCHEMBL29439748

O=C(Nc1cnccc1Cl)c1cccc(I)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.55
GSK3B P49841 1/20 0.55
POLB P06746 1/20 0.51
CACNA1B Q00975 1/20 0.51
APBA1 Q02410 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
MTOR P42345 1/20 0.49
GRM5 P41594 1/20 0.49
KDM4D Q6B0I6 1/20 0.49
KDM4C Q9H3R0 1/20 0.49
F2 P00734 1/20 0.48
LMNA P02545 1/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
KCNMA1 Q12791 1/20 0.47
MAPT P10636 1/20 0.47
BRAF P15056 2/20 0.46
TSHR P16473 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.46
NPC1 O15118 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22715632 1.00 GSK3A (0.55) GSK3AGSK3BPOLBCACNA1BAPBA1
SCHEMBL23458450 0.81 GSK3A (0.60) GSK3AGSK3BPOLBKDM4DKDM4C
SCHEMBL30785562 0.78 KMT2A (0.61) GSK3AGSK3BSMN1; SMN2KDM4DKDM4C
SCHEMBL19663017 0.77 LMNA (0.69) LMNAMEN1KMT2AMAPTTSHR
SCHEMBL17984931 0.75 CYP11B1 (0.56) GSK3AGSK3BSMN1; SMN2KDM4DKDM4C
SCHEMBL321601 0.75 CYP11B1 (0.56) GSK3AGSK3BKDM4DKDM4CLMNA
SCHEMBL3937374 0.74 CSF1R (0.80) MEN1KMT2ABRAFNPC1RAB9A
SCHEMBL19662757 0.74 BCAT2 (0.66) GRM5F2LMNABRAF
SCHEMBL7412368 0.72 ROCK2 (0.49) GSK3AGSK3BPOLBSMN1; SMN2KDM4D
SCHEMBL12685658 0.72 RHOC (0.57) POLBSMN1; SMN2GRM5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118908957-A Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-11-08 CN disclosed
CN-114222737-B Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-07-26 CN disclosed
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed
CN-114222737-A Small molecule inhibitor of NF-kB induced kinase 詹森药业有限公司 2022-03-22 CN disclosed