SCHEMBL29439813

SCHEMBL29439813

Clc1nncc2ccc(Br)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
NT5E P21589 1/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NOS1 P29475 2/20 0.36
METAP2 P50579 2/20 0.36
DYRK1A Q13627 1/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
NPM1 P06748 1/20 0.35
ALK Q9UM73 1/20 0.35
CYP2A6 P11509 1/20 0.34
BACE1 P56817 2/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17075887 1.00 HTT (0.40) HTTNT5EMEN1KMT2AMAPT
SCHEMBL396312 0.85 NOS1 (0.36) HTTNT5EMEN1KMT2AMAPT
SCHEMBL25388440 0.80 NOS1 (0.38) KMT2AMAPTKDM4EALDH1A1NOS1
SCHEMBL29677534 0.78 MEN1 (0.38) HTTMEN1KMT2AMAPTKDM4E
SCHEMBL6219191 0.78 MEN1 (0.38) HTTMEN1KMT2AMAPTKDM4E
SCHEMBL22715522 0.77 MEN1 (0.45) HTTMEN1KMT2AMAPTKDM4E
SCHEMBL23536840 0.77
SCHEMBL9998302 0.73 METAP2 (0.41) KDM4EMETAP2BACE1
SCHEMBL21432138 0.73 GABRA1 (0.42) MEN1KMT2AALDH1A1DYRK1ACYP1A2
SCHEMBL1526862 0.73 MTNR1A (0.49) MEN1KMT2AMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed