SCHEMBL29460880

SCHEMBL29460880

CCOC(=O)C1CC(C#N)(c2ccccn2)CCC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.41
NPEPPS P55786 1/20 0.39
GAA P10253 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 4/20 0.38
CASP1 P29466 2/20 0.38
HSD17B10 Q99714 2/20 0.38
HSD11B1 P28845 1/20 0.37
ALDH1A1 P00352 4/20 0.37
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PRKCA P17252 1/20 0.37
PTPN2 P17706 1/20 0.37
HTR7 P34969 1/20 0.37
HPGD P15428 3/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22538607 1.00 ADRA1A (0.41) ADRA1ANPEPPSGAAMEN1KMT2A
SCHEMBL17443847 1.00 ADRA1A (0.41) ADRA1ANPEPPSGAAMEN1KMT2A
SCHEMBL4356963 0.84 ALDH1A1 (0.45) ADRA1AMEN1KMT2AALDH1A1HTT
SCHEMBL3406286 0.80 ALDH1A1 (0.42) NPEPPSGAAKDM4ECASP1HSD17B10
SCHEMBL25001783 0.80 ALDH1A1 (0.35) NPEPPSGAAMEN1KMT2AKDM4E
SCHEMBL4253610 0.79 PKM (0.41) GAAMEN1KMT2AKDM4EHSD17B10
SCHEMBL4830643 0.77 ADORA2B (0.39) GAAMEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL3934689 0.76 PKM (0.39) GAAMEN1KMT2AKDM4EHSD17B10
SCHEMBL3931328 0.75 KDM4E (0.34) GAAMEN1KMT2AKDM4EHSD17B10
SCHEMBL3970345 0.74 PSEN1 (0.35) CASP1HSD17B10CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023081666-A1 COMPOUNDS AS CCR2 MODULATORS ARIA PHARMACEUTICALS, INC. (US) 2023-05-11 WO disclosed
CN-108602777-B 3- ((hetero-) aryl) -alkyl-8-amino-2-oxo-1, 3-aza-spiro- [4.5] -decane derivative 格吕伦塔尔有限公司 2022-05-03 CN disclosed
CN-114149413-A 3- ((hetero) aryl) -8-amino-2-oxo-1, 3-aza-spiro- [4.5] -decane derivatives 格吕伦塔尔有限公司 2022-03-08 CN disclosed