SCHEMBL2946716

SCHEMBL2946716

CC(C)(C)OC(=O)NCCc1ncc(Br)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 6/20 0.46
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
NQO2 P16083 1/20 0.40
STK17B O94768 1/20 0.40
STK17A Q9UEE5 1/20 0.40
SCN9A Q15858 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GFER P55789 1/20 0.39
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
IDO1 P14902 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
CKS1B P61024 1/20 0.36
SKP1 P63208 1/20 0.36
SKP2 Q13309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2943289 0.87 AAK1 (0.45) AAK1SCN9AIDO1CA12CA1
SCHEMBL16552184 0.85 STK17B (0.47) AAK1HTTNPSR1NQO2STK17B
SCHEMBL31362427 0.84 AAK1 (0.40) AAK1HTTNPSR1NQO2STK17B
SCHEMBL31362474 0.82 AAK1 (0.43) AAK1HTTNPSR1NQO2STK17B
SCHEMBL12476826 0.81 MTNR1B (0.40) ALDH1A1
SCHEMBL19900097 0.81 AAK1 (0.38) AAK1ALDH1A1ALOX5AP
SCHEMBL2947631 0.80 AGBL2 (0.36) ALDH1A1
SCHEMBL31569504 0.79 TDP1 (0.41) AAK1HTTNPSR1NQO2STK17B
SCHEMBL27207972 0.77 PTPN1 (0.48) AAK1IDO1
SCHEMBL27208784 0.77 PTPN1 (0.48) AAK1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396301-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS Jerini AG (DE) 2011-12-21 EP disclosed
WO-2010091876-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS JERINI AG (DE) 2010-08-19 WO disclosed