SCHEMBL29467360

SCHEMBL29467360

COCc1ccn(Cc2ccc(Cn3ccccc3=O)cc2)n1

nearest known ligand 0.50

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 20/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29324563 0.78 KLKB1 (0.59) KLKB1
SCHEMBL16578697 0.76 HDAC1 (0.50)
SCHEMBL17784852 0.76 KLKB1 (0.67) KLKB1
SCHEMBL21985437 0.76 KLKB1 (0.67) KLKB1
SCHEMBL17784845 0.76 KLKB1 (0.78) KLKB1
SCHEMBL29365582 0.76 KLKB1 (0.70) KLKB1
SCHEMBL9752787 0.75 POLB (0.63) KLKB1
SCHEMBL17685619 0.74 KLKB1 (0.46) KLKB1
Bicarbonate SCHEMBL17785352 0.72 KLKB1 (0.73) KLKB1
SCHEMBL17503935 0.72 GAA (0.53) KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464265-B1 POLYMORPHS OF N-[(3-FLUORO-4-METHOXYPYRIDIN-2-YL)METHYL]-3-(METHOXYMETHYL)-1-({4-[2-OXOPYRIDIN-1-YL)METHYL]PHENYL}METHYL)PYRAZOLE-4-CARBOXAMIDE AS KALLIKREIN INHIBITORS KALVISTA PHARMACEUTICALS LTD (GB) 2022-07-13 EP claimed
US-20250074903-A1 N-((HET)Arylmethyl)-Heteroaryl-Carboxamides Compounds As Kallikrein Inhibitors DRI UK LP (KY) 2025-03-06 US disclosed
US-20220289729-A1 N-((HET)Arylmethyl)-Heteroaryl-Carboxamides Compounds As Kallikrein Inhibitors KALVISTA PHARMACEUTICALS LTD (GB) 2022-09-15 US disclosed
EP-3982961-A1 TREATMENTS OF ANGIOEDEMA Kalvista Pharmaceuticals Limited (GB) 2022-04-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220289729-A1 N-((HET)Arylmethyl)-Heteroaryl-Carboxamides Compounds As Kallikrein Inhibitors KLKB1, BDKRB1, BDKRB2 KLKB1 1/4885
US-20250074903-A1 N-((HET)Arylmethyl)-Heteroaryl-Carboxamides Compounds As Kallikrein Inhibitors KLKB1, BDKRB1, BDKRB2 KLKB1 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.