SCHEMBL2947899

SCHEMBL2947899

N#Cc1c(Cl)cc(Cl)cc1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
KMT2A Q03164 3/20 0.33
CYP3A4 P08684 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
HPGD P15428 2/20 0.33
MEN1 O00255 2/20 0.33
TSHR P16473 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
DYRK1A Q13627 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RECQL P46063 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GPR35 Q9HC97 1/20 0.33
KDM4E B2RXH2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL952362 0.83 ALDH1A1 (0.45) ALDH1A1KMT2ACYP3A4HPGDMEN1
SCHEMBL28920176 0.78 CYP3A4 (0.41) ALDH1A1KMT2ACYP3A4L3MBTL1HPGD
SCHEMBL2429579 0.78 TRPV4 (0.43) ALDH1A1KMT2ACYP3A4L3MBTL1HPGD
SCHEMBL28031894 0.74 ALDH1A1 (0.38) ALDH1A1KMT2ACYP3A4HPGDMEN1
SCHEMBL28338346 0.74 GPR35 (0.42) ALDH1A1KMT2ACYP3A4HPGDMEN1
SCHEMBL14054812 0.74 GABRB3 (0.42) ALDH1A1KMT2ACYP3A4L3MBTL1HPGD
SCHEMBL22289598 0.74 ALDH1A1 (0.43) ALDH1A1KMT2AHPGDMEN1TP53
SCHEMBL1630139 0.73 NMT1 (0.38) ALDH1A1KMT2ACYP3A4L3MBTL1HPGD
SCHEMBL8968834 0.73 GSK3A (0.40) ALDH1A1KMT2ACYP3A4L3MBTL1HPGD
SCHEMBL967389 0.73 KDM4E (0.47) ALDH1A1KMT2ACYP3A4L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396301-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS Jerini AG (DE) 2011-12-21 EP disclosed
WO-2010091876-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS JERINI AG (DE) 2010-08-19 WO disclosed