SCHEMBL29484175

SCHEMBL29484175

COc1ccc(CNC(=S)NC(N)=O)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.71
PKM P14618 1/20 0.71
ALOX12 P18054 2/20 0.63
NPC1 O15118 1/20 0.63
CYP1A2 P05177 1/20 0.63
CYP2D6 P10635 1/20 0.63
CYP2C9 P11712 1/20 0.63
CYP2C19 P33261 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63
LMNA P02545 2/20 0.62
KDM4E B2RXH2 1/20 0.55
MAOB P27338 2/20 0.55
MAOA P21397 1/20 0.55
ATM Q13315 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
HTT P42858 1/20 0.53
GAA P10253 1/20 0.53
MAPT P10636 1/20 0.53
TDP1 Q9NUW8 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18894145 0.86 ALDH1A1 (0.73) ALDH1A1PKMALOX12NPC1CYP1A2
SCHEMBL4588187 0.84 ALDH1A1 (0.62) ALDH1A1PKMNPC1CYP2C9CYP2C19
SCHEMBL3822991 0.84 ALDH1A1 (1.00) ALDH1A1PKMALOX12LMNAMAOB
SCHEMBL11422909 0.81 ALDH1A1 (0.65) ALDH1A1PKMALOX12NPC1CYP1A2
SCHEMBL6211890 0.81 ALDH1A1 (0.80) ALDH1A1PKMALOX12LMNAKDM4E
SCHEMBL318068 0.80 ALDH1A1 (0.73) ALDH1A1PKMALOX12LMNAMAOB
SCHEMBL28230906 0.80 ALDH1A1 (0.63) ALDH1A1PKMALOX12NPC1CYP1A2
SCHEMBL21387041 0.80 ALDH1A1 (0.73) ALDH1A1PKMALOX12NPC1CYP1A2
SCHEMBL29484159 0.80 PLA2G1B (0.68) ALDH1A1ALOX12LMNAMAOBMEN1
SCHEMBL29484161 0.80 CYP2C9 (0.69) ALDH1A1ALOX12CYP2C9CYP2C19NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022055940-A1 VISTA INHIBITORS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2022-03-17 WO disclosed