SCHEMBL2948573

SCHEMBL2948573

NC(=O)c1cc2cc(C(=O)O)n(Cc3ccc(F)cc3F)c2cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 4/20 0.45
CCR9 P51686 3/20 0.43
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GPR35 Q9HC97 2/20 0.40
PTGER1 P34995 1/20 0.38
PTGDR2 Q9Y5Y4 2/20 0.37
TBXA2R P21731 1/20 0.37
ALKBH1 Q13686 1/20 0.37
JAK3 P52333 1/20 0.36
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
AURKB Q96GD4 1/20 0.36
ECE1 P42892 1/20 0.36
MAPK14 Q16539 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C8 P10632 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2945848 0.81 ALDH1A1 (0.44) KDM4EALDH1A1HSD17B10PTGER1PTGDR2
SCHEMBL2950130 0.74 MAPT (0.43) KDM4EALDH1A1HSD17B10PTGDR2ECE1
SCHEMBL2945336 0.74 PPARG (0.52) PTGER1ALKBH1
SCHEMBL6018268 0.74 CCR2 (0.59) CCR2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2943282 0.71 MAPT (0.42) KDM4EALDH1A1HSD17B10PTGDR2
SCHEMBL3033844 0.70 CCR2 (0.40) CCR2CCR9GPR35ECE1
SCHEMBL4600630 0.70 CCR2 (0.55) CCR2CCR9KDM4EALDH1A1HPGD
SCHEMBL4392732 0.70 GPR35 (0.53) CCR2CCR9GPR35
SCHEMBL9714527 0.69 GRM2 (0.43) KDM4EALDH1A1PTGER1JAK3AURKA
SCHEMBL2944416 0.69 HDAC1 (0.40) ALDH1A1PTGER1PTGDR2ECE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558611-B1 HIV-INTEGRASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND METHODS FOR THEIR USE PFIZER (US) 2010-01-06 EP claimed