SCHEMBL29488647

SCHEMBL29488647

CC(C)n1nc(Cc2c(Cl)cc(N)cc2Cl)ccc1=O

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
THRA P10827 4/20 0.32
THRB P10828 4/20 0.32
CCR2 P41597 3/20 0.32
CCR5 P51681 2/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
BPTF Q12830 1/20 0.30
ABL1 P00519 1/20 0.30
SRC P12931 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29488641 0.81 PTGDR2 (0.36) PTGDR2
SCHEMBL29488643 0.78 PTGS2 (0.38) PTGDR2
SCHEMBL29488651 0.75 DPP4 (0.37) CCR2CCR5
SCHEMBL29488656 0.74 PTGDR2 (0.53) PTGDR2
SCHEMBL24820997 0.73 MAPT (0.38) THRATHRBABL1SRC
SCHEMBL24821078 0.73 THRA (0.65) THRATHRB
SCHEMBL29488652 0.73 DPP4 (0.36) CCR2CCR5ABL1SRC
SCHEMBL29488655 0.73 GAA (0.43) SRC
SCHEMBL23370058 0.71 POLB (0.36)
SCHEMBL29488649 0.70 MAPT (0.40) THRBPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022068915-A1 6-OXO-1,6-DIHYDROPYRIDAZIN DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINE 江苏恒瑞医药股份有限公司 2022-04-07 WO disclosed