SCHEMBL29488649

SCHEMBL29488649

Nc1cc(Cl)c(Cc2ccc(=O)n(-c3cccc(F)c3)n2)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.40
MAPK14 Q16539 2/20 0.39
ADORA3 P0DMS8 3/20 0.37
ADORA2A P29274 2/20 0.37
ADORA1 P30542 1/20 0.37
P2RX7 Q99572 1/20 0.36
RXFP1 Q9HBX9 2/20 0.35
THRB P10828 1/20 0.35
AHR P35869 1/20 0.35
LMNA P02545 1/20 0.35
PTGDR2 Q9Y5Y4 3/20 0.34
FAAH O00519 1/20 0.34
MGLL Q99685 1/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
POLB P06746 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29488655 0.89 GAA (0.43) MAPTLMNAGAAHTT
SCHEMBL29488644 0.85 KMT2A (0.47) MAPTGAAHTTPOLBCYP1A2
SCHEMBL29488638 0.83 NPBWR1 (0.39) MAPTMAPK14HTT
SCHEMBL29488654 0.77 THRA (0.54) MAPTADORA3THRBLMNAHTT
SCHEMBL29488656 0.74 PTGDR2 (0.53) MAPTPTGDR2HTTCYP1A2CYP2D6
SCHEMBL29488641 0.72 PTGDR2 (0.36) MAPTPTGDR2POLBCYP1A2CYP2D6
SCHEMBL29488647 0.70 THRA (0.32) THRBPTGDR2
SCHEMBL29488643 0.70 PTGS2 (0.38) ADORA2ALMNAPTGDR2POLBCYP1A2
SCHEMBL29488651 0.69 DPP4 (0.37)
SCHEMBL29488652 0.68 DPP4 (0.36) LMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022068915-A1 6-OXO-1,6-DIHYDROPYRIDAZIN DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINE 江苏恒瑞医药股份有限公司 2022-04-07 WO disclosed