SCHEMBL29488652

SCHEMBL29488652

Nc1cc(Cl)c(Cc2ccc(=O)n(C3CCC3)n2)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.36
DPP8 Q6V1X1 2/20 0.36
PIK3CD O00329 3/20 0.34
ABL1 P00519 3/20 0.34
EGFR P00533 3/20 0.34
HCK P08631 3/20 0.34
SRC P12931 3/20 0.34
KDR P35968 3/20 0.34
PIK3CA P42336 3/20 0.34
PIK3CB P42338 3/20 0.34
MTOR P42345 3/20 0.34
PIK3CG P48736 3/20 0.34
EPHB4 P54760 3/20 0.34
PRKDC P78527 3/20 0.34
DPP9 Q86TI2 2/20 0.34
KCNH2 Q12809 3/20 0.32
PI4KB Q9UBF8 1/20 0.32
ABCB1 P08183 2/20 0.32
ADRA2A P08913 2/20 0.31
CHRM1 P11229 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29488651 0.95 DPP4 (0.37) DPP4DPP8DPP9KCNH2CCR2
SCHEMBL29488641 0.75 PTGDR2 (0.36) CYP2D6CYP3A4
SCHEMBL29488640 0.75 THRA (0.59) LMNASMN1; SMN2PDE9A
SCHEMBL29488647 0.73 THRA (0.32) ABL1SRCCCR2CCR5
SCHEMBL29488643 0.73 PTGS2 (0.38) CYP2D6LMNACYP3A4
SCHEMBL29488655 0.70 GAA (0.43) SRCLMNASMN1; SMN2
SCHEMBL29488657 0.69 THRA (0.57) LMNASMN1; SMN2
SCHEMBL24821005 0.69 MAPT (0.35) DPP4DPP8DPP9KCNH2CYP2D6
SCHEMBL29488656 0.69 PTGDR2 (0.53) CYP2D6CYP3A4SMN1; SMN2
SCHEMBL29488649 0.68 MAPT (0.40) CYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022068915-A1 6-OXO-1,6-DIHYDROPYRIDAZIN DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINE 江苏恒瑞医药股份有限公司 2022-04-07 WO disclosed