SCHEMBL2948866

SCHEMBL2948866

CS(=O)(=O)N1CCC(c2nc3c(N)nc(N)nc3[nH]2)CC1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.39
PARP2 Q9UGN5 1/20 0.36
HTR3A P46098 1/20 0.35
HTR4 Q13639 1/20 0.35
HTT P42858 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
SMYD3 Q9H7B4 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
RET P07949 1/20 0.33
KDR P35968 1/20 0.33
TP53 P04637 1/20 0.33
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32
MAPK10 P53779 1/20 0.32
KMT2A Q03164 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2950546 0.85 LMNA (0.36) PARP1HTTKMT2A
SCHEMBL15941616 0.80 MAPT (0.33) PARP1
SCHEMBL17352600 0.77 KDM4E (0.38) PARP1NPC1RAB9AHTR2B
SCHEMBL2954548 0.76 KDM4E (0.40) NPC1RAB9AHTR2B
SCHEMBL2952916 0.74
SCHEMBL2949856 0.74 DHFR (0.33)
SCHEMBL2956342 0.73 PDE4B (0.42) CCNT1CDK9
SCHEMBL2950064 0.71 HRH3 (0.36) PARP1IRAK4RETKDRMAPK8
SCHEMBL28301992 0.70 PARP1 (0.43) PARP1
SCHEMBL12095555 0.68 IDO1 (0.43) HTTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed