SCHEMBL29501419

SCHEMBL29501419

COc1ccccc1Nc1cc(C(=O)O)ncn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 1/20 0.55
TNNI3K Q59H18 1/20 0.52
NPC1 O15118 1/20 0.51
ALDH1A1 P00352 1/20 0.51
GAA P10253 1/20 0.51
MAPT P10636 1/20 0.51
RAB9A P51151 1/20 0.51
AKR1C3 P42330 2/20 0.50
AKR1C2 P52895 2/20 0.50
AURKA O14965 2/20 0.50
P4HTM Q9NXG6 1/20 0.50
EGFR P00533 4/20 0.48
ERBB3 P21860 1/20 0.48
KMO O15229 1/20 0.48
CDK4 P11802 1/20 0.47
CDK2 P24941 1/20 0.47
JAK2 O60674 1/20 0.46
JAK1 P23458 1/20 0.46
TYK2 P29597 1/20 0.46
JAK3 P52333 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25389479 1.00 MAPK10 (0.55) MAPK10TNNI3KNPC1ALDH1A1GAA
SCHEMBL30443326 0.89 MAPK10 (0.55) MAPK10TNNI3KNPC1ALDH1A1GAA
SCHEMBL25388907 0.89 MAPK10 (0.55) MAPK10TNNI3KNPC1ALDH1A1GAA
SCHEMBL3226915 0.86 S1PR1 (0.61) MAPK10TNNI3KNPC1ALDH1A1GAA
SCHEMBL13472417 0.82 KMO (0.46) EGFRERBB3KMOJAK1TYK2
SCHEMBL3227948 0.81 S1PR1 (0.61) MAPK10TNNI3KNPC1ALDH1A1GAA
SCHEMBL13300992 0.80 MAPK8 (0.62) MAPK10TNNI3KALDH1A1MAPTAKR1C3
SCHEMBL23412940 0.79 MAPT (0.55) MAPK10NPC1ALDH1A1GAAMAPT
SCHEMBL30097667 0.79 MAPT (0.55) MAPK10NPC1ALDH1A1GAAMAPT
SCHEMBL13321937 0.79 MAPK10 (0.61) MAPK10TNNI3KNPC1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116113626-A Compound with anti-tumor activity and application thereof 上海翊石医药科技有限公司 2023-05-12 CN disclosed
WO-2022048631-A1 COMPOUND HAVING ANTITUMOR ACTIVITY AND USE THEREOF 上海翊石医药科技有限公司 2022-03-10 WO disclosed