SCHEMBL2950412

SCHEMBL2950412

NNc1c(F)cc(Cl)cc1Br

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.35
MCL1 Q07820 1/20 0.33
NPC1 O15118 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM1A O60341 2/20 0.30
KDM1B Q8NB78 2/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976627 0.84 TSHR (0.35) HPGDIDO1
SCHEMBL18421429 0.84 TSHR (0.35) GAAMCL1IDO1
SCHEMBL11880006 0.76 MAPT (0.41) MAPTKMT2AGAANPC1HPGD
SCHEMBL27931109 0.75 ERN1 (0.31) MAPTKMT2A
SCHEMBL4115494 0.73 ALDH1A1 (0.41) MAPTKMT2AGAAMCL1NPC1
SCHEMBL15218429 0.72 CCR2 (0.38) MAPTKMT2AHPGDSMN1; SMN2
SCHEMBL1639839 0.71 CA1 (0.50) MAPTGAAKDM1AKDM1B
SCHEMBL17176604 0.70 GAA (0.55) MAPTKMT2AGAARAB9ASMN1; SMN2
SCHEMBL263907 0.70 PDK2 (0.37) NPC1HPGDRAB9ASMN1; SMN2KDM1A
SCHEMBL22165559 0.70 TSHR (0.35) MCL1NPC1HPGDRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396301-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS Jerini AG (DE) 2011-12-21 EP disclosed
WO-2010091876-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS JERINI AG (DE) 2010-08-19 WO disclosed