SCHEMBL29516092

SCHEMBL29516092

Cc1c(N)cncc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
F11 P03951 1/20 0.31
LPL P06858 1/20 0.30
LIPG Q9Y5X9 1/20 0.30
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20843845 1.00 F11 (0.31) F11LPLLIPGP2RX7
SCHEMBL30077920 0.79 JAK2 (0.36) LPLLIPGP2RX7
SCHEMBL9941917 0.79 LPL (0.36) LPLLIPGP2RX7
SCHEMBL28438600 0.78 UCHL1 (0.32)
SCHEMBL27191758 0.77 ESR2 (0.31)
SCHEMBL31663361 0.77 ESR2 (0.31)
SCHEMBL24667027 0.76 UCHL1 (0.35)
SCHEMBL29977339 0.76 UCHL1 (0.35)
SCHEMBL20519704 0.76 AAK1 (0.35) LPLLIPG
SCHEMBL22906863 0.75 LPL (0.36) F11LPLLIPGP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4240363-A1 7-PHENYL SUBSTITUTED 2-AMINOQUINAZOLINE INHIBITORS OF HPK1 Merck Sharp & Dohme LLC (US) 2023-09-13 EP disclosed
WO-2022098806-A1 7-PHENYL SUBSTITUTED 2-AMINOQUINAZOLINE INHIBITORS OF HPK1 MERCK SHARP & DOHME CORP. (US) 2022-05-12 WO disclosed