Synthalin

Synthalin

SCHEMBL29526432

N=C(N)NCCCCCCCCCCNC(=N)N.O=C(O)C(F)(F)F

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.48
CYP1A2 P05177 1/20 0.48
ALDH1A1 P00352 1/20 0.48
POLB P06746 1/20 0.48
ALOX15 P16050 1/20 0.44
EPHX1 P07099 1/20 0.44
CA12 O43570 1/20 0.42
CA2 P00918 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
S1PR1 P21453 4/20 0.40
S1PR3 Q99500 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6762936 0.91 SMN1; SMN2 (0.44) MEN1KMT2ASMN1; SMN2CYP1A2ALDH1A1
Agmatine SCHEMBL23364182 0.91 PAOX (0.44) MEN1KMT2ASMN1; SMN2CYP1A2ALDH1A1
Trifluoroacetic Acid SCHEMBL6761035 0.89 PRMT1 (0.48) MEN1KMT2ASMN1; SMN2CYP1A2ALDH1A1
Trifluoroacetic Acid SCHEMBL23796915 0.89 KDM4E (0.50) MEN1KMT2ASMN1; SMN2CYP1A2ALDH1A1
Trifluoroacetic Acid SCHEMBL3444104 0.89 HDAC6 (0.42) MEN1KMT2ASMN1; SMN2CYP1A2ALDH1A1
Tiformin SCHEMBL7440384 0.89 SMN1; SMN2 (0.41) MEN1KMT2ASMN1; SMN2CYP1A2ALDH1A1
Trifluoroacetic Acid SCHEMBL7439215 0.87 NPY4R (0.44) MEN1KMT2ASMN1; SMN2CYP1A2ALDH1A1
Trifluoroacetic Acid SCHEMBL4388552 0.85 KDM4E (0.45) MEN1KMT2ASMN1; SMN2CYP1A2ALDH1A1
Trifluoroacetic Acid SCHEMBL9178312 0.84 HDAC6 (0.51) MEN1KMT2ASMN1; SMN2CYP1A2ALOX15
Trifluoroacetic Acid SCHEMBL20542913 0.84 MAOA (0.57) MEN1KMT2ACA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240301429-A1 COMPOSITIONS COMPRISING SASP MODULATORS AND SENESCENCE ATTENUATORS AND USES THEREOF FOR MODULATING CELLULAR SENESCENCE RSEM, LIMITED PARTNERSHIP (CA) 2024-09-12 US claimed
US-20240301429-A1 COMPOSITIONS COMPRISING SASP MODULATORS AND SENESCENCE ATTENUATORS AND USES THEREOF FOR MODULATING CELLULAR SENESCENCE RSEM, LIMITED PARTNERSHIP (CA) 2024-09-12 US disclosed
US-12053442-B2 Methods and compositions for neuroprotection THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2024-08-06 US disclosed
US-12031137-B2 Compositions comprising SASP modulators and senescence attenuators and uses thereof for modulating cellular senescence RSEM, LIMITED PARTNERSHIP (CA) 2024-07-09 US disclosed
EP-4247405-A1 METHODS AND COMPOSITIONS FOR NEUROPROTECTION The Feinstein Institutes for Medical Research (US) 2023-09-27 EP disclosed
US-20220290122-A1 METHODS AND AGENTS FOR MODULATING MITOCHONDRIAL NAD LEVELS DAVID SABATINI, MD, PHD 2022-09-15 US disclosed
WO-2022108963-A1 METHODS AND COMPOSITIONS FOR NEUROPROTECTION THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2022-05-27 WO disclosed
US-20220151958-A1 METHODS AND COMPOSITIONS FOR NEUROPROTECTION THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2022-05-19 US disclosed
US-20220098594-A1 COMPOSITIONS COMPRISING SASP MODULATORS AND SENESCENCE ATTENUATORS AND USES THEREOF FOR MODULATING CELLULAR SENESCENCE RSEM, LIMITED PARTNERSHIP (CA) 2022-03-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12053442-B2 Methods and compositions for neuroprotection FABP7, PYGB, BDNF MEN1 4568/4885KMT2A 4321/4885SMN1; SMN2 35/4885
US-20220151958-A1 METHODS AND COMPOSITIONS FOR NEUROPROTECTION FABP7, PYGB, BDNF MEN1 4568/4885KMT2A 4321/4885SMN1; SMN2 35/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.