Davalintide

Davalintide

SCHEMBL29533482

CC(C)C[C@H](NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H]1CSSC[C@H](NC(=O)[C@@H](N)CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N1)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@H](C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O)[C@@H](C)O)[C@@H](C)O)[C@@H](C)O)[C@@H](C)O

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CALCRCALCRLRAMP1

The experimentally established mechanism targets of Davalintide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RAMP1 known ✓ O60894 1/20 0.77
CALCR known ✓ P30988 1/20 0.77
CALCRL known ✓ Q16602 1/20 0.77
RAMP2 O60895 1/20 0.77
RAMP3 O60896 1/20 0.77
NPY2R P49146 15/20 0.71
INSR P06213 1/20 0.66
PRLHR P49683 1/20 0.64
TFPI P10646 2/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Davalintide SCHEMBL29377013 0.94 RAMP1 (0.85) RAMP1RAMP2RAMP3CALCRCALCRL
SCHEMBL30078470 0.91 RAMP1 (0.91) RAMP1RAMP2RAMP3CALCRCALCRL
SCHEMBL374892 0.89 RAMP1 (0.78) RAMP1RAMP2RAMP3CALCRCALCRL
Calcitonin Salmon SCHEMBL29392873 0.89 INSR (0.64) RAMP1RAMP2RAMP3CALCRCALCRL
Calcitonin Salmon SCHEMBL269785 0.89 INSR (0.64) RAMP1RAMP2RAMP3CALCRCALCRL
SCHEMBL29511605 0.89 RAMP1 (0.71) RAMP1RAMP2RAMP3CALCRCALCRL
Amylin SCHEMBL29351499 0.88 RAMP1 (0.75) RAMP1RAMP2RAMP3CALCRCALCRL
Pramlintide SCHEMBL29355376 0.87 RAMP1 (1.00) RAMP1RAMP2RAMP3CALCRCALCRL
SCHEMBL30888738 0.87 NPY2R (0.63) RAMP1RAMP2RAMP3CALCRCALCRL
SCHEMBL29357151 0.87 RAMP1 (0.68) RAMP1RAMP2RAMP3CALCRCALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4721760-A1 COMPOSITION COMPRISING A PEPTIDE HAVING AN ISOELECTRIC POINT OF LESS THAN 6.5 AND A CO-POLYAMINO ACID BEARING CARBOXYLATE CHARGES AND HYDROPHOBIC RADICALS Adocia (FR) 2026-04-08 EP claimed
EP-4684802-A1 COMPOSITION COMPRISING A PEPTIDE HAVING AN ISOELECTRIC POINT OF LESS THAN 6.5 AND A CO-POLYAMINO ACID BEARING CARBOXYLATE CHARGES AND HYDROPHOBIC RADICALS Adocia (FR) 2026-01-28 EP claimed
WO-2025217521-A1 TREATING CHRONIC KIDNEY DISEASE WITH A COMBINATION OF A SLC6A19 INHIBITOR AND A GLP-1 AGONIST JNANA THERAPEUTICS INC. (US) 2025-10-16 WO claimed
EP-4013395-A1 COMPOSITIONS AND PARTICLES FOR PAYLOAD DELIVERY Applied Molecular Transport Inc. (US) 2022-06-22 EP claimed
CN-114555058-A Compositions and particles for payload delivery 应用分子转运公司 2022-05-27 CN claimed
WO-2026103453-A1 LONG-ACTING AMYLIN RECEPTOR AGONIST AND USE THEREOF 北京志道生物科技有限公司 2026-05-21 WO disclosed
WO-2026102089-A1 PRIME DOSE SETTING ASSEMBLY FOR INJECTION DEVICE ELI LILLY AND COMPANY (US) 2026-05-15 WO disclosed
WO-2026102086-A1 MEDICATION DELIVERY DEVICE WITH MEDICATION CARTRIDGE AND NEEDLE ASSEMBLY ELI LILLY AND COMPANY (US) 2026-05-15 WO disclosed
CN-122036914-A Long-acting amylin receptor agonist and application thereof 北京志道生物科技有限公司 2026-05-15 CN disclosed
WO-2026088071-A1 SUBSTITUTED FUSED HETEROARYL LACTAM COMPOUNDS PFIZER INC. (US) 2026-04-30 WO disclosed
US-20260116928-A1 COMPOSITIONS AND PARTICLES FOR PAYLOAD DELIVERY THORNHILL THERAPEUTICS INC (US) 2026-04-30 US disclosed
EP-4727624-A1 NEEDLE ASSEMBLY AND FLUID DELIVERY SYSTEM WITH NEEDLE ASSEMBLY Eli Lilly and Company (US) 2026-04-22 EP disclosed
US-20220380432-A1 Acylated Calcitonin Mimetics KEYBIOSCIENCE AG (CH) 2022-12-01 US disclosed
US-11504433-B2 Cholix-derived carriers for oral delivery of heterologous payload APPLIED MOLECULAR TRANSPORT INC. (US) 2022-11-22 US disclosed
US-20220288150-A1 PLANT MESSENGER PACKS ENCAPSULATING POLYPEPTIDES AND USES THEREOF FLAGSHIP PIONEERING INNOVATIONS VI, LLC 2022-09-15 US disclosed
US-20220275029-A1 COMPOSITIONS AND PARTICLES FOR PAYLOAD DELIVERY THORNHILL THERAPEUTICS, INC. 2022-09-01 US disclosed
EP-4013395-A1 COMPOSITIONS AND PARTICLES FOR PAYLOAD DELIVERY Applied Molecular Transport Inc. (US) 2022-06-22 EP disclosed
CN-114555058-A Compositions and particles for payload delivery 应用分子转运公司 2022-05-27 CN disclosed
US-20220152139-A1 PLANT MESSENGER PACKS ENCAPSULATING POLYPEPTIDES AND USES THEREOF FLAGSHIP PIONEERING INNOVATIONS VI, LLC 2022-05-19 US disclosed
US-11324833-B2 Cholix-derived carriers for oral delivery of heterologous payload APPLIED MOLECULAR TRANSPORT INC. (US) 2022-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220380432-A1 Acylated Calcitonin Mimetics CALCA, CALCRL, CALCB RAMP1 147/4885CALCR 4/4885CALCRL 2/4885
US-20260116928-A1 COMPOSITIONS AND PARTICLES FOR PAYLOAD DELIVERY SLC47A2, SLC47A1, SLC39A14 RAMP1 3260/4885CALCR 374/4885CALCRL 352/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.