SCHEMBL29538822

SCHEMBL29538822

CN1CCN(c2ccc(-c3cc4c(Br)c(Cl)cnc4n3COCC[Si](C)(C)C)cc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.40
PIM3 Q86V86 1/20 0.40
CDC7 O00311 1/20 0.37
CDK9 P50750 1/20 0.37
BRD4 O60885 9/20 0.36
ALK Q9UM73 3/20 0.36
LCK P06239 1/20 0.35
MAP4K3 Q8IVH8 1/20 0.35
MAP4K1 Q92918 1/20 0.35
FYN P06241 1/20 0.35
DGAT1 O75907 1/20 0.35
ACVRL1 P37023 1/20 0.35
ACVR1 Q04771 1/20 0.35
TNK2 Q07912 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21484370 1.00 PIM1 (0.40) PIM1PIM3CDC7CDK9BRD4
SCHEMBL21484350 0.84 PIM1 (0.40) PIM1PIM3CDC7CDK9ALK
SCHEMBL21484391 0.81 EGFR (0.44) PIM1PIM3CDK9BRD4FYN
SCHEMBL28700796 0.81 PIM1 (0.37) PIM1PIM3ALKFYNDGAT1
SCHEMBL21758128 0.75 EGFR (0.54) ALK
SCHEMBL21484332 0.73 MAPKAPK2 (0.41) BRD4
SCHEMBL21484319 0.73 EGFR (0.39) PIM1PIM3LCKMAP4K1FYN
SCHEMBL1356795 0.73 PDE1B (0.36)
SCHEMBL17289763 0.73 TBK1 (0.34) PIM1PIM3CDC7CDK9ALK
SCHEMBL1354772 0.72 DGAT1 (0.33) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110072865-B Pyrrolo-aromatic heterocyclic compounds, preparation method and medical application thereof 中国医药研究开发中心有限公司 2022-02-11 CN disclosed