SCHEMBL29544451

SCHEMBL29544451

CC(C)(C)OC(=O)n1ccc2nccc(-c3nn4c(c3Cl)C(=O)NCC4)c21

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BUB1 O43683 1/20 0.33
POLB P06746 1/20 0.32
TBK1 Q9UHD2 2/20 0.32
CNR1 P21554 1/20 0.32
MAPK1 P28482 1/20 0.31
PARP1 P09874 3/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
TNKS2 Q9H2K2 1/20 0.30
PARP2 Q9UGN5 1/20 0.30
PIM1 P11309 1/20 0.30
PIM2 Q9P1W9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29544663 0.76 RIPK3 (0.36)
SCHEMBL31440156 0.72 HSP90AA1 (0.39) BUB1POLBHSP90AA1HSP90AB1
SCHEMBL29544753 0.71 CCNC (0.36) PARP1PIM1PIM2
SCHEMBL29545041 0.71 PIM1 (0.36) MAPK1PIM1PIM2
SCHEMBL29544520 0.70 USP7 (0.38) PARP1
SCHEMBL29545095 0.70 USP7 (0.41) PARP1PIM1PIM2
SCHEMBL29544561 0.70 MET (0.34)
SCHEMBL29545167 0.70 PIK3CA (0.32) PARP1
SCHEMBL29544960 0.70 PARP1 (0.32) PARP1
SCHEMBL29544675 0.67 PIK3CA (0.40) BUB1POLBHSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022072634-A1 BICYCLIC COMPOUNDS FOR USE IN THE TREATMENT CANCER SCORPION THERAPEUTICS, INC. (US) 2022-04-07 WO disclosed