SCHEMBL29547014

SCHEMBL29547014

CC(C)(C)OC(=O)N1CC2(CC(c3c[nH]c4cc(Cl)ncc34)C2)C1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OXTR P30559 1/20 0.42
AVPR1A P37288 1/20 0.42
EHMT2 Q96KQ7 1/20 0.38
ACACB O00763 6/20 0.36
P2RX3 P56373 1/20 0.35
P2RX2 Q9UBL9 1/20 0.35
JAK1 P23458 2/20 0.35
NAMPT P43490 2/20 0.35
NR1H2 P55055 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP11B2 P19099 1/20 0.34
JAK2 O60674 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
KRAS P01116 1/20 0.34
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1F P30939 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24377843 1.00 OXTR (0.42) OXTRAVPR1AEHMT2ACACBP2RX3
SCHEMBL29546477 0.87 KDM4E (0.41) EHMT2JAK1NR1H2KDM4EJAK2
SCHEMBL24377814 0.87 KDM4E (0.41) EHMT2JAK1NR1H2KDM4EJAK2
SCHEMBL24377767 0.85 KDM4E (0.47) JAK1KDM4EJAK2TYK2JAK3
SCHEMBL29138599 0.73 OXTR (0.48) OXTRAVPR1AEHMT2ACACBNR1H2
SCHEMBL16610331 0.73 KDM4E (0.47) JAK1KDM4EJAK2TYK2JAK3
SCHEMBL4775441 0.71 GPR119 (0.46) JAK1KDM4EJAK2TYK2JAK3
SCHEMBL24377909 0.71 GABRP (0.56) JAK1CYP11B2
SCHEMBL16610447 0.71 JAK2 (0.48) JAK1KDM4EJAK2TYK2JAK3
SCHEMBL30606040 0.70 EHMT2 (0.41) OXTRAVPR1AEHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116249526-A TYK2 selective inhibitors and uses thereof 南京药石科技股份有限公司 2023-06-09 CN disclosed
WO-2022083560-A1 TYK2 SELECTIVE INHIBITOR AND USE THEREOF 南京药石科技股份有限公司 2022-04-28 WO disclosed