SCHEMBL29564442

SCHEMBL29564442

[13CH3][C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.57
KMT2A Q03164 2/20 0.54
MDM4 O15151 2/20 0.54
TP53 P04637 2/20 0.54
EPHX2 P34913 1/20 0.51
MDM2 Q00987 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26160451 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2
SCHEMBL29446045 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2
SCHEMBL29356265 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2
SCHEMBL29401309 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2
SCHEMBL119043 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2
SCHEMBL29349978 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2
SCHEMBL178736 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2
SCHEMBL29508222 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2
SCHEMBL29446029 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2
SCHEMBL119044 1.00 CASP3 (0.57) CASP3KMT2AMDM4TP53EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12618852-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2026-05-05 US disclosed
US-20260049992-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES AMBERGEN INC (US) 2026-02-19 US disclosed
US-20250369980-A1 MULTIOMIC MASS SPECTROMETRIC IMAGING OF TISSUES USING PHOTOCLEAVABLE MASS-TAG PROBES AMBEGEN INC (US) 2025-12-04 US disclosed
US-20250067751-A1 PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES AMBERGEN INC (US) 2025-02-27 US disclosed
US-12235277-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes AMBERGEN, INC. (US) 2025-02-25 US disclosed
US-12181481-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes AMBERGEN, INC. (US) 2024-12-31 US disclosed
US-12181482-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes AMBERGEN, INC. (US) 2024-12-31 US disclosed
US-20240319205-A1 Novel Photocleavable Mass-Tags for Multiplexed Mass Spectrometric Imaging of Tissues Using Biomolecular Probes AMBERGEN, INC 2024-09-26 US disclosed
US-12078639-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes AMBERGEN, INC. (US) 2024-09-03 US disclosed
US-20240264167-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES AMBERGEN, INC. 2024-08-08 US disclosed
US-20240077494-A1 Novel Photocleavable Mass-Tags for Multiplexed Mass Spectrometric Imaging of Tissues Using Biomolecular Probes AMBERGEN, INC. 2024-03-07 US disclosed
US-11906527-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes AMBERGEN, INC. (US) 2024-02-20 US disclosed
US-20230349917-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES AMBERGEN, INC. 2023-11-02 US disclosed
US-11789027-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes AMBERGEN, INC. (US) 2023-10-17 US disclosed
US-20220365097-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES AMBERGEN, INC. 2022-11-17 US disclosed
US-20220365098-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES AMBERGEN, INC 2022-11-17 US disclosed
US-20220137066-A1 PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-05-05 US disclosed
US-20220137064-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-05-05 US disclosed
US-20220137065-A1 PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-05-05 US disclosed
US-20220135518-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (16 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220365098-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES CD44, MKI67, MSH2 CASP3 2817/4885KMT2A 1336/4885MDM4 709/4885
US-12235277-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes CD44, MKI67, CD68 CASP3 2526/4885KMT2A 956/4885MDM4 754/4885
US-20230349917-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES CD44, MKI67, MSH2 CASP3 2817/4885KMT2A 1336/4885MDM4 709/4885
US-20260049992-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES MKI67, CD44, MUC1 CASP3 1417/4885KMT2A 1222/4885MDM4 700/4885
US-12618852-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes CD44, CD68, EPCAM CASP3 2522/4885KMT2A 2197/4885MDM4 921/4885
US-20240264167-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES CD44, MKI67, MSH2 CASP3 2817/4885KMT2A 1336/4885MDM4 709/4885
US-11906527-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes CD44, MKI67, CD68 CASP3 2526/4885KMT2A 956/4885MDM4 754/4885
US-12181481-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes CD44, MKI67, CD68 CASP3 2526/4885KMT2A 956/4885MDM4 754/4885
US-20220365097-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES CD44, MKI67, MSH2 CASP3 2817/4885KMT2A 1336/4885MDM4 709/4885
US-20240319205-A1 Novel Photocleavable Mass-Tags for Multiplexed Mass Spectrometric Imaging of Tissues Using Biomolecular Probes CD44, MKI67, MSH2 CASP3 2817/4885KMT2A 1336/4885MDM4 709/4885
US-11789027-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes MKI67, MSH2, MSH6 CASP3 1752/4885KMT2A 389/4885MDM4 114/4885
US-20220135518-A1 NOVEL PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES CD44, MKI67, MSH2 CASP3 2817/4885KMT2A 1336/4885MDM4 709/4885
US-20250067751-A1 PHOTOCLEAVABLE MASS-TAGS FOR MULTIPLEXED MASS SPECTROMETRIC IMAGING OF TISSUES USING BIOMOLECULAR PROBES CD44, MKI67, CD68 CASP3 2526/4885KMT2A 956/4885MDM4 754/4885
US-20240077494-A1 Novel Photocleavable Mass-Tags for Multiplexed Mass Spectrometric Imaging of Tissues Using Biomolecular Probes CD44, MKI67, MSH2 CASP3 2817/4885KMT2A 1336/4885MDM4 709/4885
US-12181482-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes MKI67, MSH2, MSH6 CASP3 1752/4885KMT2A 389/4885MDM4 114/4885
US-12078639-B2 Photocleavable mass-tags for multiplexed mass spectrometric imaging of tissues using biomolecular probes CD44, MKI67, CD68 CASP3 2526/4885KMT2A 956/4885MDM4 754/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.