SCHEMBL29566635

SCHEMBL29566635

Clc1cncc(CN2CCNCC2)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.54
CHRNA4 P43681 3/20 0.54
SIGMAR1 Q99720 1/20 0.51
CHRNA1 P02708 1/20 0.49
CHRNA7 P36544 1/20 0.49
CXCR4 P61073 12/20 0.47
MEN1 O00255 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
ADRA2C P18825 1/20 0.47
CCR2 P41597 1/20 0.47
CXCL12 P48061 1/20 0.47
BLM P54132 1/20 0.47
KMT2A Q03164 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
PTPN11 Q06124 1/20 0.45
SOS1 Q07889 1/20 0.43
ADRB2 P07550 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22422495 1.00 CHRNB2 (0.54) CHRNB2CHRNA4SIGMAR1CHRNA1CHRNA7
SCHEMBL626347 0.80 L3MBTL1 (0.61) SIGMAR1CXCR4MEN1CHRM2CHRM1
SCHEMBL27969917 0.80 CHRNB2 (0.47) CHRNB2CHRNA4SIGMAR1CXCR4MEN1
SCHEMBL13770498 0.80 CXCR4 (0.49) SIGMAR1CXCR4MEN1CHRM2CHRM1
SCHEMBL18390568 0.80 MC4R (0.51) SIGMAR1TDP1
SCHEMBL4757486 0.80 SIGMAR1 (0.47) SIGMAR1CXCR4MEN1CHRM2CHRM1
Hydrochloric Acid SCHEMBL17062037 0.79 L3MBTL1 (0.59) SIGMAR1CXCR4MEN1CHRM2CHRM1
SCHEMBL17929340 0.79 CXCR4 (0.68) CHRNB2CHRNA4SIGMAR1CXCR4MEN1
SCHEMBL17828171 0.78 ACHE (0.54) HRH3
SCHEMBL26665904 0.77 SIGMAR1 (0.55) CHRNB2CHRNA4SIGMAR1CXCR4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114380825-B Substituted pyrazole condensed ring derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2024-02-13 CN disclosed
CN-112771043-B Substituted pyrazole condensed ring derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2023-04-28 CN disclosed
CN-114380825-A Substituted pyrazole fused ring derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2022-04-22 CN disclosed