SCHEMBL2958

SCHEMBL2958

N#Cc1ccccc1-c1ccc(CNCCCOCc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.48
UGCG Q16739 1/20 0.48
GBA2 Q9HCG7 1/20 0.48
FFAR1 O14842 1/20 0.45
AKR1B1 P15121 1/20 0.45
ESR2 Q92731 1/20 0.43
EGLN1 Q9GZT9 1/20 0.42
BCHE P06276 2/20 0.42
SCN8A Q9UQD0 2/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2739 0.93 FFAR1 (0.46) GBA1UGCGGBA2FFAR1AKR1B1
SCHEMBL2083 0.84 SCN8A (0.46) FFAR1AKR1B1ESR2SCN8AMEN1
SCHEMBL6961295 0.84 FFAR1 (0.55) GBA1UGCGGBA2FFAR1AKR1B1
SCHEMBL6960223 0.83 GBA1 (0.54) GBA1UGCGGBA2FFAR1AKR1B1
SCHEMBL2405 0.82 DRD4 (0.50) FFAR1AKR1B1ESR2BCHESCN8A
SCHEMBL6960030 0.82 ESR2 (0.59) GBA1UGCGGBA2FFAR1AKR1B1
SCHEMBL6961121 0.81 GBA1 (0.56) GBA1UGCGGBA2FFAR1AKR1B1
SCHEMBL6952546 0.81 FFAR1 (0.57) GBA1UGCGGBA2FFAR1AKR1B1
SCHEMBL15341674 0.80 MAOA (0.62) BCHESCN8ATSHRMEN1KMT2A
SCHEMBL2401 0.80 ESR2 (0.50) FFAR1AKR1B1ESR2TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed