SCHEMBL2401

SCHEMBL2401

N#Cc1ccccc1-c1ccc(CNCCCCO)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.50
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PDCD1 Q15116 1/20 0.47
CD274 Q9NZQ7 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
MAOA P21397 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
MYC P01106 1/20 0.43
WDR5 P61964 1/20 0.43
HRH4 Q9H3N8 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
CHRM2 P08172 1/20 0.42
MME P08473 1/20 0.42
FFAR1 O14842 1/20 0.42
AKR1B1 P15121 1/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2694 0.99 ESR2 (0.49) ESR2MEN1KMT2APDCD1CD274
SCHEMBL6606543 0.86 HRH4 (0.54) ESR2MEN1KMT2APDCD1CD274
SCHEMBL2405 0.83 DRD4 (0.50) ESR2MEN1KMT2AMAOACYP1A2
SCHEMBL6606339 0.83 ESR2 (0.49) ESR2MEN1KMT2APDCD1CD274
SCHEMBL2083 0.83 SCN8A (0.46) ESR2MEN1KMT2APDCD1CD274
SCHEMBL6957868 0.81 ESR2 (0.57) ESR2MYCWDR5MMEFFAR1
SCHEMBL2958 0.80 GBA1 (0.48) ESR2MEN1KMT2AMAOACYP1A2
SCHEMBL6961869 0.80 ESR2 (0.56) ESR2MYCWDR5MMEFFAR1
SCHEMBL2545 0.80 L3MBTL1 (0.47) ESR2MEN1KMT2APDCD1CD274
SCHEMBL6957117 0.79 ESR2 (0.59) ESR2MYCWDR5MMEFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed