SCHEMBL29580189

SCHEMBL29580189

Clc1ccc(CNc2ccccn2)c(Cl)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.69
GAA P10253 1/20 0.68
KDM4E B2RXH2 2/20 0.62
GPR39 O43194 2/20 0.62
TSHR P16473 1/20 0.58
SLC2A1 P11166 1/20 0.54
HPGD P15428 2/20 0.54
ALDH1A1 P00352 1/20 0.54
CXCR4 P61073 1/20 0.53
FABP1 P07148 1/20 0.51
FABP6 P51161 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
MEN1 O00255 1/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 1/20 0.49
LMNA P02545 1/20 0.48
NPC1 O15118 1/20 0.48
MITF O75030 1/20 0.48
TP53 P04637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29579974 0.88 POLB (0.74) POLBGAAKDM4EGPR39TSHR
SCHEMBL18947190 0.85 NPSR1 (0.66) POLBGAAKDM4EGPR39HPGD
SCHEMBL29579757 0.85 GAA (0.57) POLBGAAKDM4EGPR39HPGD
SCHEMBL29579775 0.83 ALDH1A1 (0.65) POLBGAAKDM4EGPR39HPGD
SCHEMBL14321086 0.81 GAA (0.53) POLBGAAKDM4EGPR39TSHR
SCHEMBL14321655 0.81 GAA (0.53) POLBGAAKDM4EGPR39TSHR
SCHEMBL27299487 0.81 GAA (0.53) POLBGAAKDM4EGPR39TSHR
SCHEMBL29557927 0.77 GPR39 (1.00) GPR39SLC2A1
SCHEMBL29580040 0.77 KDM4E (1.00) POLBGAAKDM4EGPR39TSHR
SCHEMBL14980562 0.77 KDM4E (1.00) POLBGAAKDM4EGPR39TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113651811-B Isoxazole-containing pyridopyrimidone compound and preparation method and application thereof 贵州大学 2022-06-07 CN disclosed