SCHEMBL29587458

SCHEMBL29587458

COc1ccc(-c2ccc3c(c2)OC(C(=O)NOC2CCCCO2)CC3)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.40
NFKB1 P19838 2/20 0.39
NFKB2 Q00653 2/20 0.39
RELA Q04206 2/20 0.39
NPC1 O15118 3/20 0.39
ALDH1A1 P00352 3/20 0.39
RAB9A P51151 3/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
HDAC3 O15379 3/20 0.38
HDAC1 Q13547 3/20 0.38
HDAC2 Q92769 3/20 0.38
LMNA P02545 3/20 0.38
MAPK1 P28482 2/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPT P10636 1/20 0.37
ADORA3 P0DMS8 1/20 0.36
FFAR1 O14842 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29587460 0.86 SLC6A3 (0.39) NFKB1NFKB2RELAHDAC3HDAC1
SCHEMBL29587203 0.84 PPARG (0.39) HPGDNFKB1NFKB2RELAALDH1A1
SCHEMBL29587169 0.82 HDAC3 (0.45) HPGDNFKB1NFKB2RELAALDH1A1
SCHEMBL29587175 0.82 FAAH (0.36) NPC1RAB9AHDAC3HDAC1HDAC2
SCHEMBL29586866 0.82 LMNA (0.42) HPGDNPC1ALDH1A1RAB9ALMNA
SCHEMBL29587290 0.82 HDAC3 (0.51) NFKB1NFKB2RELAALDH1A1RAB9A
SCHEMBL29588212 0.81 RAB9A (0.48) HPGDNFKB1NFKB2RELANPC1
SCHEMBL29586783 0.80 HDAC3 (0.44) HPGDNFKB1NFKB2RELAHDAC3
SCHEMBL29586900 0.80 HDAC3 (0.44) HPGDNFKB1NFKB2RELAHDAC3
SCHEMBL29587076 0.79 SLC6A3 (0.39) NFKB1NFKB2RELANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022120048-A1 HDAC INHIBITORS UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2022-06-09 WO disclosed