SCHEMBL29601464

SCHEMBL29601464

Cn1cc(-c2nc(-c3ccc(Cl)cc3)cnc2NNC(N)=S)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.44
FGFR3 P22607 1/20 0.44
CSF1R P07333 3/20 0.40
AURKB Q96GD4 2/20 0.40
AURKA O14965 1/20 0.40
MAPK1 P28482 4/20 0.37
S1PR2 O95136 2/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
CHEK1 O14757 2/20 0.37
KDM1A O60341 1/20 0.37
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
MAPKAPK2 P49137 1/20 0.36
PARP1 P09874 1/20 0.35
CCNT1 O60563 1/20 0.35
CCNB2 O95067 1/20 0.35
CCNE2 O96020 1/20 0.35
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24327324 0.83 FGFR3 (0.50) KDRFGFR3CSF1RAURKBAURKA
SCHEMBL28724019 0.82 FGFR3 (0.51) KDRFGFR3CSF1RAURKBAURKA
SCHEMBL24327827 0.77 FGFR3 (0.53) KDRFGFR3CSF1RAURKBAURKA
SCHEMBL29498949 0.76 FGFR3 (0.56) KDRFGFR3CSF1RAURKBAURKA
SCHEMBL24327350 0.76 FGFR3 (0.56) KDRFGFR3CSF1RAURKBAURKA
SCHEMBL24328692 0.76 EPHB4 (0.40) FGFR3AURKBMAPK1CHEK1CDK2
SCHEMBL24328703 0.75 FGFR3 (0.51) KDRFGFR3CSF1RAURKBAURKA
SCHEMBL24327370 0.75 FGFR3 (0.51) KDRFGFR3CSF1RAURKBAURKA
SCHEMBL24327347 0.74 KDR (0.53) KDRFGFR3CSF1RAURKBAURKA
SCHEMBL29498933 0.74 KDR (0.53) KDRFGFR3CSF1RAURKBAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114369097-A Heteroaromatic AhR inhibitors 山东轩竹医药科技有限公司 2022-04-19 CN disclosed