SCHEMBL29601993

SCHEMBL29601993

C[C@H](N)C(=O)N[C@@H](CCCCN)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CO)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NTSR2 O95665 2/20 0.40
NTSR1 P30989 2/20 0.40
NAALAD2 Q9Y3Q0 1/20 0.39
NRP1 O14786 2/20 0.38
OPRM1 P35372 3/20 0.37
CTSB P07858 1/20 0.37
CPB2 Q96IY4 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29752649 0.90 NTSR2 (0.43) NTSR2NTSR1NAALAD2NRP1OPRM1
SCHEMBL31114334 0.87 OPRM1 (0.55) NTSR2NTSR1OPRM1CTSB
SCHEMBL30612366 0.87 NAALAD2 (0.44) NTSR2NTSR1NAALAD2OPRM1CPB2
SCHEMBL29601866 0.84 OPRM1 (0.51) NTSR2NTSR1OPRM1
SCHEMBL31114523 0.84 NRP1 (0.44) NTSR2NTSR1NAALAD2NRP1OPRM1
SCHEMBL31114333 0.82 NTSR2 (0.51) NTSR2NTSR1OPRM1CTSB
SCHEMBL30361658 0.82 NTSR2 (0.43) NTSR2NTSR1NRP1CTSBCPB2
SCHEMBL31114385 0.81 OPRM1 (0.57) NTSR2NTSR1OPRM1
SCHEMBL31114378 0.81 NAALAD2 (0.45) NAALAD2NRP1OPRM1CPB2
SCHEMBL30877896 0.81 NAALAD2 (0.42) NAALAD2CPB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4665372-A1 NEW MULTI-FUNCTIONAL OLIGOPEPTIDES EnliTISA (Shanghai) Pharmaceutical Co., Ltd. (CN) 2025-12-24 EP claimed
US-20250066417-A9 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2025-02-27 US claimed
WO-2024169972-A1 NEW MULTI-FUNCTIONAL OLIGOPEPTIDES Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2024-08-22 WO claimed
US-20240182520-A1 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS ENLITISA SHANGHAI PHARMACEUTICAL CO LTD (CN) 2024-06-06 US claimed
US-20240165247-A1 NEW PEPTIDE CONJUGATES Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2024-05-23 US claimed
US-20240124521-A1 NEW PEPTIDES JIANGYIN USUN PHARMACEUTICAL CO., LTD. (CN) 2024-04-18 US claimed
EP-4308167-A1 NEW PEPTIDE CONJUGATES EnliTISA (Shanghai) Pharmaceutical Co., Ltd. (CN) 2024-01-24 EP claimed
EP-4308584-A1 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS EnliTISA (Shanghai) Pharmaceutical Co., Ltd. (CN) 2024-01-24 EP claimed
CN-117425498-A Novel peptide conjugates 艾缇亚(上海)制药有限公司 2024-01-19 CN claimed
CN-117396491-A Novel peptide-based diagnostic and therapeutic agents 艾缇亚(上海)制药有限公司 2024-01-12 CN claimed
US-20230113836-A1 NEW CONJUGATES OF PEPTIDES AND POLYSACCHARIDE Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2023-04-13 US claimed
EP-4069713-A1 NEW CONJUGATES OF PEPTIDES AND POLYSACCHARIDE EnliTISA (Shanghai) Pharmaceutical Co., Ltd. (CN) 2022-10-12 EP claimed
WO-2022194239-A1 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2022-09-22 WO claimed
WO-2022193186-A1 NEW DIAGNOSTIC AND THERAPEUTIC AGENTS JIANGYIN USUN PHARMACEUTICAL CO., LTD. (CN) 2022-09-22 WO claimed
WO-2022193185-A1 NEW CONJUGATES JIANGYIN USUN PHARMACEUTICAL CO., LTD. (CN) 2022-09-22 WO claimed
WO-2022194238-A1 NEW PEPTIDE CONJUGATES Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2022-09-22 WO claimed
CN-114929283-A Novel conjugates of peptides and polysaccharides 艾缇亚(上海)制药有限公司 2022-08-19 CN claimed
EP-4028409-A1 NEW PEPTIDES Jiangyin Usun Pharmaceutical Co., Ltd. (CN) 2022-07-20 EP claimed
CN-114375298-A Novel peptides 江阴贝瑞森制药有限公司 2022-04-19 CN claimed
US-12612430-B2 Peptides Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2026-04-28 US disclosed
EP-4665372-A1 NEW MULTI-FUNCTIONAL OLIGOPEPTIDES EnliTISA (Shanghai) Pharmaceutical Co., Ltd. (CN) 2025-12-24 EP disclosed
US-20250066417-A9 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2025-02-27 US disclosed
WO-2024169972-A1 NEW MULTI-FUNCTIONAL OLIGOPEPTIDES Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2024-08-22 WO disclosed
US-20240182520-A1 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS ENLITISA SHANGHAI PHARMACEUTICAL CO LTD (CN) 2024-06-06 US disclosed
US-20240165247-A1 NEW PEPTIDE CONJUGATES Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2024-05-23 US disclosed
US-20240124521-A1 NEW PEPTIDES JIANGYIN USUN PHARMACEUTICAL CO., LTD. (CN) 2024-04-18 US disclosed
EP-4308167-A1 NEW PEPTIDE CONJUGATES EnliTISA (Shanghai) Pharmaceutical Co., Ltd. (CN) 2024-01-24 EP disclosed
EP-4308584-A1 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS EnliTISA (Shanghai) Pharmaceutical Co., Ltd. (CN) 2024-01-24 EP disclosed
CN-117425498-A Novel peptide conjugates 艾缇亚(上海)制药有限公司 2024-01-19 CN disclosed
CN-117396491-A Novel peptide-based diagnostic and therapeutic agents 艾缇亚(上海)制药有限公司 2024-01-12 CN disclosed
US-20230113836-A1 NEW CONJUGATES OF PEPTIDES AND POLYSACCHARIDE Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2023-04-13 US disclosed
EP-4069713-A1 NEW CONJUGATES OF PEPTIDES AND POLYSACCHARIDE EnliTISA (Shanghai) Pharmaceutical Co., Ltd. (CN) 2022-10-12 EP disclosed
WO-2022194239-A1 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2022-09-22 WO disclosed
WO-2022193186-A1 NEW DIAGNOSTIC AND THERAPEUTIC AGENTS JIANGYIN USUN PHARMACEUTICAL CO., LTD. (CN) 2022-09-22 WO disclosed
WO-2022193185-A1 NEW CONJUGATES JIANGYIN USUN PHARMACEUTICAL CO., LTD. (CN) 2022-09-22 WO disclosed
WO-2022194238-A1 NEW PEPTIDE CONJUGATES Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2022-09-22 WO disclosed
CN-114929283-A Novel conjugates of peptides and polysaccharides 艾缇亚(上海)制药有限公司 2022-08-19 CN disclosed
EP-4028409-A1 NEW PEPTIDES Jiangyin Usun Pharmaceutical Co., Ltd. (CN) 2022-07-20 EP disclosed
CN-114375298-A Novel peptides 江阴贝瑞森制药有限公司 2022-04-19 CN disclosed
CN-114375298-A Novel peptides 江阴贝瑞森制药有限公司 2022-04-19 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230113836-A1 NEW CONJUGATES OF PEPTIDES AND POLYSACCHARIDE DSG1, HBG1, IDUA NTSR2 3899/4885NTSR1 3426/4885NAALAD2 709/4885
US-20250066417-A9 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS NGLY1, YBX1, VIP NTSR2 1057/4885NTSR1 892/4885NAALAD2 597/4885
US-20240182520-A1 NEW PEPTIDE-BASED DIAGNOSTIC AND THERAPEUTIC AGENTS NGLY1, YBX1, VIP NTSR2 1057/4885NTSR1 892/4885NAALAD2 597/4885
US-12612430-B2 Peptides CUTA, VIP, COL14A1 NTSR2 1049/4885NTSR1 1080/4885NAALAD2 358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.