552-02 Free Base

552-02 Free Base

SCHEMBL29615808

CS(=O)(=O)O.N=C(NCCCCc1ccc(OCC(O)CO)cc1)NC(=O)c1nc(Cl)c(N)nc1N

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of 552-02 Free Base. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SCNN1A P37088 18/20 0.67
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
552-02 Free Base SCHEMBL15092803 1.00 SCNN1A (0.67) SCNN1AKCNH2
552-02 Free Base SCHEMBL9913757 0.97 SCNN1A (0.71) SCNN1A
552-02 Free Base SCHEMBL2015162 0.97 SCNN1A (0.71) SCNN1A
552-02 Free Base SCHEMBL9913774 0.97 SCNN1A (0.71) SCNN1A
552-02 Free Base SCHEMBL19348088 0.96 SCNN1A (0.70) SCNN1A
SCHEMBL916347 0.94 SCNN1A (0.67) SCNN1A
SCHEMBL14268270 0.91 SCNN1A (0.60) SCNN1AKCNH2
SCHEMBL10028716 0.91 SCNN1A (0.60) SCNN1AKCNH2
SCHEMBL14268271 0.91 SCNN1A (0.60) SCNN1AKCNH2
SCHEMBL10110701 0.90 SCNN1A (0.62) SCNN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4713056-A1 DEVICE FOR PROVIDING CONTINUED BREATH GUIDANCE, METHOD OF OPERATING AN INHALATION DEVICE, INHALATION DEVICE AND INHALATION DEVICE SYSTEM FOR PROVIDING INHALATION PROCESS/BREATH GUIDING Pari Medical Holding GmbH (DE) 2026-03-25 EP disclosed
EP-4712837-A1 METHOD OF OPERATING AN INHALATION DEVICE, INHALATION DEVICE, INHALATION DEVICE SYSTEM FOR PROVIDING INHALATION PROCESS FEEDBACK AND DEVICE FOR PROVIDING FEEDBACK GUIDANCE Pari Medical Holding GmbH (DE) 2026-03-25 EP disclosed
US-12544520-B2 Aerosol delivery device and method of operating the aerosol delivery device PARI PHARMA GMBH (DE) 2026-02-10 US disclosed
EP-4659255-A1 MEDICAL EVALUATION METHOD, AEROSOL NEBULIZER AND MEDICAL EVALUATION SYSTEM Pari Medical Holding GmbH (DE) 2025-12-10 EP disclosed
WO-2024236034-A1 DEVICE FOR PROVIDING CONTINUED BREATH GUIDANCE, METHOD OF OPERATING AN INHALATION DEVICE, INHALATION DEVICE AND INHALATION DEVICE SYSTEM FOR PROVIDING INHALATION PROCESS/BREATH GUIDING PARI MEDICAL HOLDING GMBH (DE) 2024-11-21 WO disclosed
WO-2024236057-A1 METHOD OF OPERATING AN INHALATION DEVICE, INHALATION DEVICE, INHALATION DEVICE SYSTEM FOR PROVIDING INHALATION PROCESS FEEDBACK AND DEVICE FOR PROVIDING FEEDBACK GUIDANCE PARI MEDICAL HOLDING GMBH (DE) 2024-11-21 WO disclosed
WO-2024160951-A1 MEDICAL EVALUATION METHOD, AEROSOL NEBULIZER AND MEDICAL EVALUATION SYSTEM PARI MEDICAL HOLDING GMBH (DE) 2024-08-08 WO disclosed
EP-4259607-A1 BENZIMIDAZOLE DERIVATIVES FOR TREATING RESPIRATORY DISEASE TMEM16A LIMITED (GB) 2023-10-18 EP disclosed
EP-4082023-A1 CONTROL DEVICE FOR AEROSOL NEBULIZER SYSTEM PARI Pharma GmbH (DE) 2022-11-02 EP disclosed
WO-2022123314-A1 BENZIMIDAZOLE DERIVATIVES FOR TREATING RESPIRATORY DISEASE TMEM16A LIMITED (GB) 2022-06-16 WO disclosed
CN-110214141-B Benzodiazolium compounds as ENaC inhibitors 企业治疗学有限公司 2022-05-31 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12544520-B2 Aerosol delivery device and method of operating the aerosol delivery device VAPA, VAPB, PIEZO1 SCNN1A 452/4885KCNH2 411/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.