SCHEMBL29615833

SCHEMBL29615833

c1cncc(CN2CCN3CCOCC3C2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV6 Q9H1D0 5/20 0.54
CHRNB2 P17787 1/20 0.50
CHRNA4 P43681 1/20 0.50
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 4/20 0.43
TDP1 Q9NUW8 2/20 0.43
KMT2A Q03164 1/20 0.43
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.42
HPGD P15428 1/20 0.42
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL310319 0.84 SIGMAR1 (0.49) TRPV6ALDH1A1DRD4
SCHEMBL1189566 0.84 SIGMAR1 (0.49) TRPV6ALDH1A1DRD4
SCHEMBL29615692 0.81 TRPV6 (0.62) TRPV6CHRNB2CHRNA4OPRM1OPRD1
SCHEMBL29615698 0.81 TRPV6 (0.62) TRPV6CHRNB2CHRNA4OPRM1OPRD1
SCHEMBL20528276 0.79 PIK3CA (0.39) TRPV6
SCHEMBL18201926 0.79 PIK3CA (0.39) TRPV6
SCHEMBL31329931 0.78 TRPV6 (0.80) TRPV6CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL4970159 0.76 CHRNB2 (0.72) TRPV6CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL21553313 0.76 CNR2 (0.41) TRPV6
SCHEMBL16026435 0.74 CHRNB2 (0.85) TRPV6CHRNB2CHRNA4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11351170-B2 Substituted pyrimidines as CDK4/6 inhibitors BEIJING XUANYI PHARMASCIENCES CO., LTD. (CN) 2022-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11351170-B2 Substituted pyrimidines as CDK4/6 inhibitors CDK4, CDK6, CDK2 TRPV6 3973/4885CHRNB2 3875/4885CHRNA4 3227/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.