SCHEMBL29615698

SCHEMBL29615698

c1cncc(CN2CCN3CCCC3C2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV6 Q9H1D0 4/20 0.62
CHRNB2 P17787 1/20 0.57
CHRNA4 P43681 1/20 0.57
ALDH1A1 P00352 4/20 0.53
MAPT P10636 1/20 0.53
HTT P42858 1/20 0.53
KDM4E B2RXH2 5/20 0.52
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49
OPRK1 P41145 1/20 0.49
ROCK2 O75116 1/20 0.48
CCR2 P41597 1/20 0.48
ROCK1 Q13464 1/20 0.48
MAPK1 P28482 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
CASP1 P29466 1/20 0.46
CASP4 P49662 1/20 0.46
CASP5 P51878 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29615692 1.00 TRPV6 (0.62) TRPV6CHRNB2CHRNA4ALDH1A1MAPT
SCHEMBL31329931 0.84 TRPV6 (0.80) TRPV6CHRNB2CHRNA4ALDH1A1KDM4E
SCHEMBL23225374 0.83 ALDH1A1 (0.58) TRPV6ALDH1A1KDM4EMAPK1MEN1
SCHEMBL21216229 0.83 ALDH1A1 (0.58) TRPV6ALDH1A1KDM4EMAPK1MEN1
SCHEMBL28283653 0.82 CHRNB2 (0.71) TRPV6CHRNB2CHRNA4ALDH1A1MAPT
SCHEMBL29615833 0.81 TRPV6 (0.54) TRPV6CHRNB2CHRNA4ALDH1A1MAPT
SCHEMBL938061 0.79 CHRNB2 (0.61) TRPV6CHRNB2CHRNA4ALDH1A1MAPT
SCHEMBL5091037 0.79 SIGMAR1 (0.54) TRPV6ALDH1A1KDM4EMAPK1MEN1
SCHEMBL12250 0.78 CHRNB2 (0.65) TRPV6CHRNB2CHRNA4ALDH1A1MAPT
SCHEMBL12449679 0.78 CHRNB2 (0.65) TRPV6CHRNB2CHRNA4ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11351170-B2 Substituted pyrimidines as CDK4/6 inhibitors BEIJING XUANYI PHARMASCIENCES CO., LTD. (CN) 2022-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11351170-B2 Substituted pyrimidines as CDK4/6 inhibitors CDK4, CDK6, CDK2 TRPV6 3973/4885CHRNB2 3875/4885CHRNA4 3227/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.