SCHEMBL29616670

SCHEMBL29616670

Cc1ccc(C(F)(F)F)c(-c2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.46
HDAC7 Q8WUI4 1/20 0.44
PSMB5 P28074 1/20 0.42
AR P10275 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
PDK2 Q15119 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
MAPT P10636 2/20 0.40
S1PR1 P21453 2/20 0.39
S1PR3 Q99500 1/20 0.39
MAOB P27338 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
PLK1 P53350 1/20 0.39
ELANE P08246 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23149011 1.00 HSD11B1 (0.46) HSD11B1HDAC7PSMB5ARPTGDR2
SCHEMBL5114438 0.87 AR (0.51) HSD11B1ARPDK2MAOBCYP3A4
SCHEMBL4637120 0.85 AKR1C3 (0.51) HSD11B1HDAC7PSMB5ARPDK2
SCHEMBL26375405 0.83 KIF11 (0.42) HSD11B1ARAKR1C3AKR1C2MAPT
SCHEMBL26375409 0.82 HSD11B1 (0.50) HSD11B1ARPDK2CYP1A2CYP3A4
SCHEMBL26375407 0.82 NFE2L2 (0.45) ARAKR1C3AKR1C2MAPTCYP1A2
SCHEMBL16363206 0.81 KIF11 (0.51) HSD11B1ARPDK2AKR1C3AKR1C2
SCHEMBL12439813 0.81 CYP46A1 (0.46) HSD11B1MAPTS1PR1S1PR3KDM4E
SCHEMBL29890189 0.81 HSD11B1 (0.48) HSD11B1PSMB5ARPTGDR2AKR1C3
SCHEMBL28838153 0.81 HSD11B1 (0.48) HSD11B1PSMB5ARPTGDR2AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114401968-A Novel heterocyclic monoacylglycerol lipase (MAGL) inhibitors 豪夫迈·罗氏有限公司 2022-04-26 CN disclosed