SCHEMBL29616972

SCHEMBL29616972

N#Cc1cccc(-c2ncnc3[nH]ncc23)c1F

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 8/20 0.46
MAPK1 P28482 2/20 0.41
HTT P42858 2/20 0.41
MKNK1 Q9BUB5 1/20 0.41
PTK2 Q05397 1/20 0.40
RET P07949 1/20 0.39
PI4KA P42356 1/20 0.39
XDH P47989 1/20 0.39
PI4K2B Q8TCG2 1/20 0.39
PI4K2A Q9BTU6 1/20 0.39
PI4KB Q9UBF8 1/20 0.39
ADORA2A P29274 1/20 0.39
RPS6KB1 P23443 3/20 0.38
TRPA1 O75762 1/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
PRKCQ Q04759 1/20 0.37
MAP4K1 Q92918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29761062 0.87 TRPA1 (0.47) LRRK2MAPK1MKNK1PTK2RET
SCHEMBL29761065 0.77 LRRK2 (0.41) LRRK2MAPK1HTTMKNK1PTK2
SCHEMBL29761000 0.76 RET (0.41) LRRK2MAPK1HTTMKNK1PTK2
SCHEMBL3677097 0.74 L3MBTL1 (0.46) LRRK2MAPK1HTTMKNK1PTK2
SCHEMBL29761017 0.73 LRRK2 (0.45) LRRK2
SCHEMBL16906740 0.71 PTK2 (0.42) HTTPTK2RPS6KB1TRPA1LMNA
SCHEMBL29761064 0.68 ADORA2A (0.51) ADORA2ATRPA1
SCHEMBL19575560 0.68 RET (0.40) LRRK2MAPK1HTTMKNK1PTK2
SCHEMBL3260282 0.68 BTK (0.47) LRRK2MAPK1PTK2RETPI4KA
SCHEMBL745097 0.68 RET (0.43) LRRK2MAPK1PTK2RETPI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116425756-A Adenosine receptor antagonist compounds and uses thereof 日东制药株式会社 2023-07-14 CN disclosed
CN-114829363-A Adenosine receptor antagonist compounds 日东制药株式会社 2022-07-29 CN disclosed
WO-2022107044-A1 PREVENTION AND/OR TREATMENT OF CNS DISORDERS ILDONG PHARMACEUTICAL CO., LTD. (KR) 2022-05-27 WO disclosed