SCHEMBL29761065

SCHEMBL29761065

N#Cc1cccnc1-c1ncnc2[nH]ncc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.41
RET P07949 1/20 0.41
PI4KA P42356 1/20 0.41
XDH P47989 1/20 0.41
PI4K2B Q8TCG2 1/20 0.41
PI4K2A Q9BTU6 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAPK1 P28482 2/20 0.40
METAP2 P50579 2/20 0.40
PDPK1 O15530 1/20 0.39
LMNA P02545 2/20 0.38
CHEK1 O14757 1/20 0.38
AURKA O14965 1/20 0.38
HTT P42858 1/20 0.38
CSF1R P07333 1/20 0.37
PTK2 Q05397 1/20 0.37
CNR2 P34972 1/20 0.37
SLC29A1 Q99808 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29761062 0.82 TRPA1 (0.47) LRRK2RETPI4KAXDHPI4K2B
SCHEMBL29761000 0.80 RET (0.41) LRRK2RETPI4KAXDHPI4K2B
SCHEMBL29616972 0.77 LRRK2 (0.46) LRRK2RETPI4KAXDHPI4K2B
SCHEMBL31267979 0.74 CNR2 (0.49) LRRK2HTTCNR2MAPTHDAC1
SCHEMBL29761078 0.72 L3MBTL1 (0.52) LRRK2RETPI4KAXDHPI4K2B
SCHEMBL3677097 0.71 L3MBTL1 (0.46) LRRK2RETPI4KAXDHPI4K2B
SCHEMBL29761040 0.71 RET (0.41) LRRK2RETPI4KAXDHPI4K2B
SCHEMBL5419659 0.71 ROCK2 (0.44) LRRK2RETPI4KAXDHPI4K2B
SCHEMBL29761041 0.70 AKT2 (0.43) LRRK2PI4KAXDHPI4K2BPI4K2A
SCHEMBL29993245 0.69 XDH (0.55) LRRK2RETPI4KAXDHPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116425756-A Adenosine receptor antagonist compounds and uses thereof 日东制药株式会社 2023-07-14 CN disclosed
CN-114829363-A Adenosine receptor antagonist compounds 日东制药株式会社 2022-07-29 CN disclosed