SCHEMBL29617710

SCHEMBL29617710

N#Cc1cccc(C(=O)NCc2ccc(B(O)O)cc2)c1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.55
CHRM3 P20309 1/20 0.52
GAA P10253 1/20 0.49
P4HB P07237 1/20 0.48
EPHX2 P34913 2/20 0.48
ENPP2 Q13822 1/20 0.48
HDAC2 Q92769 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
MAOA P21397 1/20 0.47
GPR139 Q6DWJ6 1/20 0.46
NR1H4 Q96RI1 1/20 0.46
ROCK2 O75116 1/20 0.46
GSK3B P49841 1/20 0.46
VNN1 O95497 3/20 0.46
NAMPT P43490 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17339504 1.00 TRPV1 (0.55) TRPV1CHRM3GAAP4HBEPHX2
SCHEMBL17339214 0.89 CHRM3 (0.56) CHRM3GAAEPHX2ENPP2HDAC2
SCHEMBL17142140 0.85 HDAC2 (0.64) CHRM3GAAEPHX2HDAC2HDAC8
SCHEMBL5091359 0.84 CHRM3 (0.54) CHRM3GAAEPHX2HDAC2HDAC8
SCHEMBL7233161 0.84 CHRM3 (0.54) CHRM3GAAEPHX2HDAC2HDAC8
SCHEMBL17339532 0.84 EPHX2 (0.67) TRPV1EPHX2ENPP2HDAC6MAOA
SCHEMBL7989764 0.83 GAA (0.53) CHRM3GAAEPHX2HDAC2HDAC8
SCHEMBL7985996 0.83 GAA (0.56) CHRM3GAAVNN1
SCHEMBL28146231 0.83 CHRM3 (0.55) CHRM3GAAEPHX2HDAC2HDAC8
SCHEMBL17339264 0.82 VNN1 (0.49) CHRM3GAAP4HBEPHX2ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685516-A Pyrazolopyrimidine derivatives as BTK inhibitors for the treatment of cancer 洛克索肿瘤学股份有限公司 2022-07-01 CN disclosed
CN-108431007-B Pyrazolopyrimidine derivatives as BTK inhibitors for the treatment of cancer 洛克索肿瘤学股份有限公司 2022-06-07 CN disclosed