SCHEMBL29617795

SCHEMBL29617795

COc1ccc(Cl)cc1C(=O)NCc1ccc(B(O)O)cc1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.62
DNMT3A Q9Y6K1 1/20 0.59
PPARA Q07869 1/20 0.58
HDAC1 Q13547 2/20 0.55
HDAC6 Q9UBN7 2/20 0.55
NLRP3 Q96P20 3/20 0.54
HPGD P15428 1/20 0.52
TSHR P16473 1/20 0.52
RECQL P46063 1/20 0.52
ALDH1A1 P00352 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17339437 1.00 LMNA (0.62) LMNADNMT3APPARAHDAC1HDAC6
SCHEMBL17339271 0.90 AKR1B1 (0.54) LMNADNMT3APPARAHPGDALDH1A1
SCHEMBL23657593 0.90 LMNA (0.72) LMNADNMT3APPARAHDAC1HDAC6
SCHEMBL17339512 0.88 HPGD (0.55) PPARAHPGDALDH1A1
SCHEMBL11516368 0.87 LMNA (0.68) LMNADNMT3APPARAHDAC1HDAC6
SCHEMBL29471048 0.85 PTGER4 (0.54) LMNAPPARAHPGDALDH1A1
SCHEMBL17339505 0.85 PTGER4 (0.54) LMNAPPARAHPGDALDH1A1
SCHEMBL11356211 0.84 LMNA (0.64) LMNADNMT3APPARAHDAC1HDAC6
SCHEMBL11464602 0.84 PTGER4 (0.69) LMNADNMT3APPARAHDAC1HDAC6
SCHEMBL11706059 0.83 DNMT3A (0.72) LMNADNMT3APPARAHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685516-A Pyrazolopyrimidine derivatives as BTK inhibitors for the treatment of cancer 洛克索肿瘤学股份有限公司 2022-07-01 CN disclosed
CN-108431007-B Pyrazolopyrimidine derivatives as BTK inhibitors for the treatment of cancer 洛克索肿瘤学股份有限公司 2022-06-07 CN disclosed