SCHEMBL23657593

SCHEMBL23657593

COc1ccc(Cl)cc1C(=O)NCc1ccc(Cl)cc1

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.72
PPARA Q07869 1/20 0.69
DNMT3A Q9Y6K1 1/20 0.67
HDAC1 Q13547 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
NLRP3 Q96P20 3/20 0.60
HPGD P15428 1/20 0.58
ALDH1A1 P00352 1/20 0.58
TSHR P16473 1/20 0.58
RECQL P46063 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11516368 0.94 LMNA (0.68) LMNAPPARADNMT3AHDAC1HDAC6
SCHEMBL11464602 0.91 PTGER4 (0.69) LMNAPPARADNMT3AHDAC1HDAC6
SCHEMBL11356211 0.91 LMNA (0.64) LMNAPPARADNMT3AHDAC1HDAC6
SCHEMBL29617795 0.90 LMNA (0.62) LMNAPPARADNMT3AHDAC1HDAC6
SCHEMBL11706059 0.90 DNMT3A (0.72) LMNAPPARADNMT3AHDAC1HDAC6
SCHEMBL17339437 0.90 LMNA (0.62) LMNAPPARADNMT3AHDAC1HDAC6
SCHEMBL23042429 0.89 PPARA (0.64) LMNAPPARADNMT3AHPGDALDH1A1
SCHEMBL11488803 0.89 PPARA (0.67) LMNAPPARADNMT3AHDAC1HDAC6
SCHEMBL14507293 0.88 LMNA (0.60) LMNAPPARADNMT3AHDAC1HDAC6
SCHEMBL11445600 0.86 LMNA (0.63) LMNAPPARADNMT3AHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210220408-A1 ARYL HYDROCARBON RECEPTOR ANTAGONISTS AND METHODS OF USE EDIGENE BIOTECHNOLOGY, INC. (CN) 2021-07-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210220408-A1 ARYL HYDROCARBON RECEPTOR ANTAGONISTS AND METHODS OF USE AHR, ARNT, ARSA LMNA 3403/4885PPARA 50/4885DNMT3A 3082/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.