SCHEMBL29618319

SCHEMBL29618319

N#Cc1ccc2c(c1)CC(F)(F)C2

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PNMT P11086 6/20 0.46
DRD2 P14416 4/20 0.46
DRD3 P35462 4/20 0.46
KDM1A O60341 2/20 0.41
CXCR5 P32302 3/20 0.39
PDK2 Q15119 1/20 0.36
TRPA1 O75762 1/20 0.35
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
TYRO3 Q06418 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12715536 0.80 POLB (0.46) PNMTDRD2DRD3KDM1ACXCR5
SCHEMBL29506141 0.74 PNMT (0.49) PNMTDRD2DRD3KDM1A
SCHEMBL22789739 0.74 PNMT (0.49) PNMTDRD2DRD3KDM1A
SCHEMBL24878784 0.72 DRD2 (0.43) PNMTDRD2DRD3KDM1A
SCHEMBL27795984 0.72 CXCR5 (0.47) PNMTDRD2DRD3KDM1ACXCR5
SCHEMBL6739755 0.72
SCHEMBL24878782 0.71 HRH3 (0.42) PNMTDRD2DRD3KDM1ACXCR5
SCHEMBL18710410 0.71 EPAS1 (0.30)
SCHEMBL24275671 0.70 TDP2 (0.41) PNMTKDM1A
Bromide SCHEMBL17202846 0.70 PNMT (0.52) PNMTDRD2DRD3KDM1ATRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022121805-A1 FUSED RING COMPOUND AS NAV1.8 INHIBITOR AND USE THEREOF 成都康弘药业集团股份有限公司 2022-06-16 WO disclosed
CN-114591293-A Fused ring compound as Nav1.8 inhibitor and application thereof 成都康弘药业集团股份有限公司 2022-06-07 CN disclosed