SCHEMBL29620496

SCHEMBL29620496

CC(=O)c1ccc(Br)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
HPGD P15428 1/20 0.47
MAPT P10636 2/20 0.44
PKM P14618 2/20 0.44
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
MAOB P27338 3/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
S100A4 P26447 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KIF11 P52732 2/20 0.42
CYP2A6 P11509 1/20 0.41
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL333891 1.00 ALDH1A1 (0.47) ALDH1A1HPGDMAPTPKMCES2
SCHEMBL381027 0.83 NPC1 (0.44) ALDH1A1HPGDMAPTPKMCES2
SCHEMBL16955913 0.83 SLC6A4 (0.39) ALDH1A1HPGDMAPTCES2CES1
SCHEMBL286942 0.81 HTT (0.53) HPGDMAPTCES2CES1MAOB
SCHEMBL30523532 0.81 HTT (0.53) HPGDMAPTCES2CES1MAOB
SCHEMBL29669896 0.80 CES2 (0.67) MAPTPKMCES2CES1MAOB
SCHEMBL75801 0.80 CES2 (0.67) MAPTPKMCES2CES1MAOB
SCHEMBL3022646 0.80 MAPT (0.47) ALDH1A1HPGDMAPTPKMS100A4
SCHEMBL356759 0.79 KIF11 (0.49) CES2CES1MAOBHDAC1HDAC6
SCHEMBL321581 0.79 CES2 (0.43) ALDH1A1MAPTCES2CES1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248510-B Salts of 2-fluoro-N-methyl-4- [7- (quinolin-6-ylmethyl) imidazo [1,2-b ] [1,2,4] triazin-2-yl ] benzamide and methods for preparing same 因西特控股公司 2025-01-17 CN disclosed
CN-119233976-A Modulators of c-MYC mRNA translation and their use in the treatment of cancer 艾尼莫生物科技公司 2024-12-31 CN disclosed
CN-119176772-A Compound with Mrgpr X receptor inhibition effect and application thereof 博济医药科技股份有限公司 2024-12-24 CN disclosed
CN-118679160-A BRM targeting compounds and related methods of use 阿维纳斯运营公司 2024-09-20 CN disclosed
CN-118488950-A ENPP1 inhibitors 上海齐鲁制药研究中心有限公司 2024-08-13 CN disclosed
CN-114555597-B Isocitrate Dehydrogenase (IDH) inhibitors 浙江迈同生物医药有限公司 2024-06-04 CN disclosed
EP-4298098-A1 SULFONYL BENZAMIDE DERIVATIVES AS BCL-2 INHIBITORS Ascentage Pharma (Suzhou) Co., Ltd. (CN) 2024-01-03 EP disclosed
EP-3802550-B1 NOVEL BENZIMIDAMIDES COMPOUNDS COMPRISING AN OXABORININ RING INST NAT SANTE RECH MED (FR) 2023-12-27 EP disclosed
CN-114835704-B Sulfonylbenzamide derivatives as BCL-2 inhibitors 苏州亚盛药业有限公司 2023-10-27 CN disclosed
CN-110177783-B Hormone receptor modulators for the treatment of metabolic conditions and disorders 阿德利克斯股份有限公司 2023-06-06 CN disclosed
CN-112236433-B Novel compounds 国家医疗保健研究所 2023-04-04 CN disclosed
CN-115361948-A Methods and compositions for inhibiting dihydroorotate dehydrogenase 俄亥俄州国家创新基金会 2022-11-18 CN disclosed
EP-4041732-A1 ISO-CITRATE DEHYDROGENASE (IDH) INHIBITOR ZHEJIANG METON PHARMACEUTICAL CO., LTD (CN) 2022-08-17 EP disclosed
CN-114874143-A Regulator containing pyrazole derivatives, preparation method and application thereof 上海翰森生物医药科技有限公司 2022-08-09 CN disclosed
WO-2022161496-A1 SULFONYL BENZAMIDE DERIVATIVES AS BCL-2 INHIBITORS ASCENTAGE PHARMA (SUZHOU) CO., LTD. (CN) 2022-08-04 WO disclosed
CN-114835704-A Sulfonylbenzamide derivatives as BCL-2 inhibitors 苏州亚盛药业有限公司 2022-08-02 CN disclosed
CN-114555597-A Isocitrate Dehydrogenase (IDH) inhibitors 浙江迈同生物医药有限公司 2022-05-27 CN disclosed