SCHEMBL29623796

SCHEMBL29623796

CCNc1cccc(C(N)=O)c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.47
MKNK1 Q9BUB5 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45
PARP1 P09874 2/20 0.42
HSD17B10 Q99714 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
USP2 O75604 1/20 0.41
CASP1 P29466 1/20 0.41
BRCA1 P38398 1/20 0.41
CASP7 P55210 1/20 0.41
AGTR1 P30556 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13073788 0.84 NPC1 (0.53) KDM4EHSD17B10ALDH1A1HPGDNPC1
SCHEMBL3441356 0.84 AGTR1 (0.54) KDM4EMKNK1MKNK2ALDH1A1HPGD
Hydrochloric Acid SCHEMBL5389527 0.82 AGTR1 (0.53) KDM4EMKNK1MKNK2ALDH1A1HPGD
SCHEMBL13450268 0.80 KDM4E (0.50) KDM4EPARP1HSD17B10ALDH1A1HPGD
SCHEMBL31481384 0.80 KDM4E (0.50) KDM4EPARP1HSD17B10ALDH1A1HPGD
SCHEMBL29623849 0.80 BTK (0.57) KDM4EHSD17B10ALDH1A1HPGDNPC1
SCHEMBL15387043 0.79 KDM4E (0.49) KDM4EPARP1HSD17B10ALDH1A1HPGD
Formic Acid SCHEMBL5388605 0.78 MEN1 (0.49) KDM4EMKNK1MKNK2HSD17B10ALDH1A1
SCHEMBL7868859 0.78 MEN1 (0.40) KDM4EHSD17B10ALDH1A1HPGDNPC1
SCHEMBL7259307 0.78 FABP4 (0.54) MKNK1MKNK2MEN1KMT2AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113024516-B Double-target PARP/EZH2 inhibitor, preparation method and application 中国药科大学 2022-05-17 CN disclosed