SCHEMBL29628340

SCHEMBL29628340

C=Cc1ccc(C(F)(F)F)nc1OC

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.35
MBOAT4 Q96T53 1/20 0.35
HSD17B10 Q99714 2/20 0.33
PDE4B Q07343 4/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32
TUBB3 Q13509 1/20 0.32
TUBB2A Q13885 1/20 0.32
TUBB8 Q3ZCM7 1/20 0.32
TUBA3E Q6PEY2 1/20 0.32
TUBA1A Q71U36 1/20 0.32
TUBA1C Q9BQE3 1/20 0.32
TUBB6 Q9BUF5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30971780 0.83 PDE4B (0.39) NT5EMBOAT4HSD17B10PDE4BCYP1A2
SCHEMBL2131813 0.83 PDE4B (0.39) NT5EMBOAT4HSD17B10PDE4BCYP1A2
SCHEMBL14844545 0.77 MBOAT4 (0.37) NT5EMBOAT4HSD17B10PDE4BCYP1A2
SCHEMBL2132119 0.75 PRMT1 (0.43) CYP1A2CYP2C9CYP2C19HPGDNPSR1
SCHEMBL2132111 0.75 PRMT1 (0.43) CYP1A2CYP2C9CYP2C19HPGDNPSR1
SCHEMBL24468866 0.74 TRPV4 (0.32) NT5E
SCHEMBL12093699 0.74 MBOAT4 (0.38) MBOAT4HSD17B10PDE4BTUBB4ATUBB
SCHEMBL2614964 0.74 MBOAT4 (0.40) MBOAT4HSD17B10PDE4BTUBB4ATUBB
SCHEMBL19172629 0.73 MBOAT4 (0.42) MBOAT4HSD17B10PDE4BTUBB4ATUBB
SCHEMBL15201463 0.73 ULK1 (0.39) NT5EMBOAT4HSD17B10PDE4BTUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3997096-A1 NEW HETEROCYCLIC COMPOUNDS F. Hoffmann-La Roche AG (CH) 2022-05-18 EP disclosed